SCHEMBL9836619

SCHEMBL9836619

c1ccc2c(c1)Cc1cccnc1C(NCCN1CCOCC1)O2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
HPGDS O60760 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MITF O75030 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
SMARCA2 P51531 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
LTA4H P09960 2/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836563 0.91 ADRA2C (0.36) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL9836638 0.77 CYP2C19 (0.41) KDM4EMEN1KMT2ALMNAHPGD
SCHEMBL9835190 0.76 HTR1A (0.35) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL9837035 0.75 OPRL1 (0.42) CXCR4LMNALTA4HCYP3A4CYP2D6
SCHEMBL9834580 0.75 HRH1 (0.36) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL9835645 0.74 ALDH1A1 (0.37) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL9836246 0.70 MTNR1A (0.40) L3MBTL1KDM4ELMNAALDH1A1TSHR
SCHEMBL9836609 0.70 MEN1 (0.41) CXCR4L3MBTL1KDM4ENPC1RAB9A
SCHEMBL9834815 0.68 CHRM2 (0.42) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL11011112 0.68 CHRM2 (0.34) CXCR4L3MBTL1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP claimed
US-4547496-A Antiulcer [1] benzepino[3,4-b]pyridine and compositions KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-10-15 US claimed
EP-0129879-A2 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-02 EP claimed