SCHEMBL9836747

SCHEMBL9836747

CCNC(=O)N(CC)C1Oc2ccccc2Cc2cccnc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
TSHR P16473 2/20 0.36
HTT P42858 2/20 0.36
HPGD P15428 3/20 0.34
MAPK1 P28482 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
CHIA Q9BZP6 1/20 0.33
LMNA P02545 2/20 0.32
MEN1 O00255 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836558 0.78 MEN1 (0.33) GAAL3MBTL1TSHRHTTHPGD
SCHEMBL9836832 0.72 ALDH1A1 (0.34) GAAL3MBTL1TSHRHTTMAPK1
Diethylamine SCHEMBL9836584 0.72 HTT (0.37) GAAL3MBTL1TSHRHTTLMNA
SCHEMBL9836739 0.70 TSHR (0.36) GAAL3MBTL1TSHRHTTHPGD
SCHEMBL9835190 0.68 HTR1A (0.35) HTT
SCHEMBL9837005 0.68 MAOA (0.41) HTTMEN1KMT2ASMN1; SMN2
SCHEMBL9836246 0.68 MTNR1A (0.40) GAAL3MBTL1TSHRHTTHDAC3
SCHEMBL9835645 0.67 ALDH1A1 (0.37) GAATSHRHTT
SCHEMBL9835181 0.66 MAOA (0.41) TSHR
SCHEMBL9837246 0.66 MAOA (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP claimed
US-4547496-A Antiulcer [1] benzepino[3,4-b]pyridine and compositions KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-10-15 US claimed
EP-0129879-A2 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-02 EP claimed