SCHEMBL9836832

SCHEMBL9836832

CCN(CC)CC(=O)NC1Oc2ccccc2Cc2cccnc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
MAPT P10636 3/20 0.34
RAB9A P51151 1/20 0.34
GFER P55789 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
GAA P10253 3/20 0.34
HTT P42858 2/20 0.34
TSHR P16473 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
P2RX7 Q99572 1/20 0.34
LMNA P02545 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPK1 P28482 1/20 0.33
MC4R P32245 1/20 0.33
SCN4A P35499 1/20 0.33
MC3R P41968 1/20 0.33
HTR3A P46098 1/20 0.33
SCN5A Q14524 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836246 0.83 MTNR1A (0.40) ALDH1A1MAPTGAAHTTTSHR
Diethylamine SCHEMBL9836584 0.81 HTT (0.37) ALDH1A1GAAHTTTSHRL3MBTL1
SCHEMBL9835190 0.79 HTR1A (0.35) ALDH1A1HTTLTA4H
SCHEMBL9835645 0.77 ALDH1A1 (0.37) ALDH1A1GAAHTTTSHRLTA4H
SCHEMBL9836747 0.72 GAA (0.36) GAAHTTTSHRL3MBTL1LMNA
SCHEMBL9836638 0.72 CYP2C19 (0.41) ALDH1A1GAATSHRLMNA
SCHEMBL9837005 0.71 MAOA (0.41) HTTP2RX7SMN1; SMN2
SCHEMBL9836562 0.70 P2RX7 (0.36) ALDH1A1MAPTNPSR1GAAP2RX7
SCHEMBL9834580 0.70 HRH1 (0.36) TDP1TSHRCYP3A4BLM
SCHEMBL9836558 0.69 MEN1 (0.33) ALDH1A1GAAHTTTSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP claimed
US-4547496-A Antiulcer [1] benzepino[3,4-b]pyridine and compositions KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-10-15 US claimed
EP-0129879-A2 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-02 EP claimed
EP-0129879-A2 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-02 EP disclosed