SCHEMBL9837429

SCHEMBL9837429

CC(C)(Cc1c[nH]c2ccccc12)N1C[C@@H](COc2cccc3[nH]ccc23)OC1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 9/20 0.41
SLC6A4 P31645 3/20 0.41
CYP2D6 P10635 4/20 0.40
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SLC22A1 O15245 1/20 0.37
GRM2 Q14416 3/20 0.36
TACR1 P25103 1/20 0.35
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
ADRA1D P25100 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
ADRA1A P35348 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10559798 0.81 TACR1 (0.40) HTR1ASLC6A4CYP2D6DRD2DRD4
SCHEMBL10558466 0.78 NR3C1 (0.40) CYP2D6MEN1KMT2AGRM2TACR1
SCHEMBL11220571 0.75 HTR1A (0.45) HTR1ACYP2D6DRD4DRD3MEN1
SCHEMBL11482581 0.72 CA2 (0.47) MEN1KMT2AGRM2MAPK1
SCHEMBL9835784 0.70 PKM (0.43) HTR1ASLC6A4DRD2DRD4DRD3
SCHEMBL9837332 0.70 PKM (0.43) HTR1ASLC6A4DRD2DRD4DRD3
SCHEMBL10558635 0.70 PKM (0.43) HTR1ASLC6A4DRD2DRD4DRD3
SCHEMBL9835778 0.70 PKM (0.43) HTR1ASLC6A4DRD2DRD4DRD3
SCHEMBL9837336 0.70 PKM (0.43) HTR1ASLC6A4DRD2DRD4DRD3
SCHEMBL11215201 0.70 HTR1B (0.44) HTR1ACYP2D6DRD4DRD3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0251938-B1 STEREOSPECIFIC PROCESS FOR THE SYNTHESIS OF INDOLE DERIVATIVES SANOFI (FR) 1991-11-06 EP claimed
EP-0240107-B1 THIANAPHTHENE DERIVATIVES, THEIR PRODUCTION AND USE Sankyo Company Limited (JP) 1991-08-21 EP disclosed
US-5021444-A Anticoagulants SANKYO COMPANY LIMITED (JP) 1991-06-04 US disclosed
US-4847272-A ANTICOAGULANTS SANKYO COMPANY LIMITED (JP) 1989-07-11 US disclosed
US-4806655-A Process for the stereospecific synthesis of indole derivatives SOCIETE ANONYME: SANOFI (FR) 1989-02-21 US disclosed