SCHEMBL9844766

SCHEMBL9844766

Cn1cc(CCc2ccc(C(=O)O)cc2)c2c(N)ncnc21

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.46
LCK P06239 1/20 0.46
TEK Q02763 1/20 0.46
EP300 Q09472 3/20 0.45
MBOAT4 Q96T53 1/20 0.45
XDH P47989 1/20 0.42
SRC P12931 3/20 0.41
RET P07949 2/20 0.40
EIF2AK3 Q9NZJ5 3/20 0.39
EGFR P00533 2/20 0.38
FYN P06241 1/20 0.38
ABL1 P00519 1/20 0.37
CDK1 P06493 1/20 0.37
ABL2 P42684 1/20 0.37
SLC16A3 O15427 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844770 0.87 EP300 (0.49) KDREP300SRCRETEGFR
SCHEMBL27709073 0.83 MBOAT4 (0.50) EP300MBOAT4SLC16A3
SCHEMBL9844798 0.81 PTGER1 (0.42) KDRLCKTEKEP300SLC16A3
SCHEMBL9844757 0.80 DHFR (0.55)
SCHEMBL9844775 0.75 DHFR (0.43)
SCHEMBL9844769 0.75 DHFR (0.43)
SCHEMBL14647492 0.74 ADORA2A (0.43) EIF2AK3
SCHEMBL9844768 0.72 TBXAS1 (0.39) EP300MBOAT4
SCHEMBL18100426 0.67 ADK (0.55) KDRLCKSRCRETEIF2AK3
SCHEMBL22676116 0.66 KDR (0.47) KDRLCKTEKXDHSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed