SCHEMBL9844822

SCHEMBL9844822

CN1CC(CCCc2ccc(C(=O)O)cc2)c2c(O)nc(N)nc21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 2/20 0.37
RARB P10826 6/20 0.37
HRH1 P35367 1/20 0.36
KCNH2 Q12809 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RARA P10276 1/20 0.36
MAPT P10636 1/20 0.36
MTOR P42345 1/20 0.36
KMT2A Q03164 1/20 0.36
EP300 Q09472 2/20 0.36
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER3 P43115 1/20 0.35
PTGER2 P43116 1/20 0.35
TLR7 Q9NYK1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844816 0.80 DHFR (0.42) ALDH1A1
SCHEMBL9844754 0.78 ATIC (0.51)
SCHEMBL8997177 0.77 NOS1 (0.39) TBXAS1RARBMEN1ALDH1A1RARA
SCHEMBL8567466 0.70 MTR (0.41) RARBMAPTKMT2A
SCHEMBL9844790 0.69 EP300 (0.38) HRH1MEN1MAPTKMT2AEP300
SCHEMBL8997209 0.69 CYP4A11 (0.43) ALDH1A1EP300TLR7
SCHEMBL9338914 0.67 CYP2D6 (0.56) RARBMEN1ALDH1A1RARAMAPT
SCHEMBL9341089 0.67 CYP2D6 (0.53) TBXAS1RARBMEN1ALDH1A1RARA
SCHEMBL9844768 0.66 TBXAS1 (0.39) TBXAS1RARBMEN1ALDH1A1RARA
SCHEMBL9343568 0.66 CYP2D6 (0.55) RARBMEN1ALDH1A1RARAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed