SCHEMBL9846701

SCHEMBL9846701

CC1CCN(C2=NC(C)(C)Oc3ccccc32)C1=O

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.33
PLA2G1B P04054 1/20 0.33
ATG4B Q9Y4P1 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
PER2 O15055 3/20 0.32
BACE1 P56817 3/20 0.31
CTSD P07339 2/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
MAP3K5 Q99683 2/20 0.31
HDAC4 P56524 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HRH4 Q9H3N8 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846679 0.84 SIGMAR1 (0.33) ATMSIGMAR1PER2ADRA1DADRA1A
SCHEMBL9846720 0.83 PBRM1 (0.37) BACE1CTSD
SCHEMBL9846780 0.77 PDK2 (0.39) HDAC4HDAC8
SCHEMBL9846762 0.70 OPRM1 (0.33)
SCHEMBL9372567 0.69 ADK (0.32) ATMSIGMAR1HRH4
SCHEMBL9846735 0.69 IDH1 (0.33) BACE1CTSDADRA1AHRH4
SCHEMBL9846707 0.69 ACHE (0.35)
SCHEMBL9373066 0.67 ADK (0.33)
SCHEMBL13194218 0.65 BACE1 (0.48) BACE1
SCHEMBL266004 0.65 MEN1 (0.50) SIGMAR1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0450487-A1 Benzoxazine derivatives, method for their preparation and their use for treating or prophylaxis of diseases HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-09 EP disclosed