SCHEMBL9848672

SCHEMBL9848672

CC(C)[C@H](NC(=O)C(Cc1ccccc1)Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(=O)OC(C)(C)C)C(=O)N[C@H]([C]=O)CC(C)(C)C)C(C)C

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 11/20 0.47
REN P00797 3/20 0.42
PSEN1 P49768 2/20 0.41
PSEN2 P49810 2/20 0.41
APH1B Q8WW43 2/20 0.41
NCSTN Q92542 2/20 0.41
APH1A Q96BI3 2/20 0.41
PSENEN Q9NZ42 2/20 0.41
APP P05067 1/20 0.41
CTSD P07339 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9848617 0.83 BACE1 (0.38) BACE1RENCTSD
SCHEMBL9848673 0.80 BACE1 (0.53) BACE1CTSD
SCHEMBL9848705 0.75 BACE1 (0.43) BACE1RENCTSD
SCHEMBL9848692 0.74 LTA4H (0.54)
SCHEMBL9848678 0.73 BACE1 (0.42) BACE1RENCTSD
SCHEMBL11199973 0.72 CTSS (0.54) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL8528279 0.72 PSEN1 (0.57) BACE1RENPSEN1PSEN2APH1B
SCHEMBL2185519 0.71 CTSC (0.54) BACE1CTSD
SCHEMBL17456239 0.70 OPRD1 (0.55)
SCHEMBL9848649 0.69 BACE1 (0.55) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438873-A1 Inhibitor of ribonucleotide reductase of herpes viruses MERCK & CO. INC. (US) 1991-07-31 EP disclosed