SCHEMBL9864432

SCHEMBL9864432

[NH]C(=O)c1ccc(Br)cc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.52
CES2 O00748 2/20 0.52
GALR3 O60755 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
HPGD P15428 1/20 0.52
CASP1 P29466 1/20 0.52
CYP2C19 P33261 1/20 0.52
GSTA1 P08263 1/20 0.44
MAPT P10636 2/20 0.44
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 1/20 0.43
ALOX12 P18054 1/20 0.43
RAB9A P51151 1/20 0.43
DGAT1 O75907 1/20 0.42
ERN1 O75460 1/20 0.41
BCL2 P10415 1/20 0.39
MCL1 Q07820 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6154796 0.83 ALOX15 (0.69) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL13740129 0.83 DGAT1 (0.62) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL467470 0.80 ALDH1A1 (0.61) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL29433676 0.78 MAOA (0.58) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL28768383 0.78 MAOA (0.58) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL55915 0.78 MAOA (0.58) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL2956396 0.78 ALOX15 (0.52) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL20505340 0.77 CES2 (0.55) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL25666683 0.77 MAPT (0.54) ALOX15CES2GALR3CYP1A2CYP2C9
SCHEMBL3526226 0.77 GAA (0.55) ALOX15CES2GALR3CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011938-A Antimicrobials ELI LILLY AND COMPANY (US) 1991-04-30 US disclosed
US-4940718-A BACTERICIDES ELI LILLY AND COMPANY (US) 1990-07-10 US disclosed
US-4795815-A BACTERICIDES, MICROBIOCIDES ELI LILLY AND COMPANY (US) 1989-01-03 US disclosed
US-4716232-A 1-(vinyl phosphonate adduct) pyrazolidinones ELI LILLY AND COMPANY (US) 1987-12-29 US disclosed
EP-0202794-A1 7-Substituted-2,3-(Dihydro) bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-11-26 EP disclosed
EP-0202046-A1 7-Substituted bicyclic pyrazolidinones ELI LILLY AND COMPANY (US) 1986-11-20 EP disclosed