SCHEMBL9865584

SCHEMBL9865584

O=C(CCNC(=O)c1cccc(NC(=O)c2ccc(CNC(=O)OCc3ccccc3)cc2)c1)OCc1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.60
HDAC1 Q13547 3/20 0.55
HDAC2 Q92769 2/20 0.55
HDAC3 O15379 1/20 0.55
PAX8 Q06710 1/20 0.51
NR1H4 Q96RI1 2/20 0.50
LMNA P02545 1/20 0.50
MAPK1 P28482 1/20 0.50
KDM1A O60341 1/20 0.48
MAOA P21397 1/20 0.48
KDM1B Q8NB78 1/20 0.48
RCOR1 Q9UKL0 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
HTT P42858 1/20 0.48
MMP2 P08253 1/20 0.48
MMP9 P14780 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867345 0.94 NAMPT (0.52) NAMPTPAX8NR1H4LMNAMAPK1
SCHEMBL9864590 0.87 PAX8 (0.52) NAMPTPAX8NR1H4LMNAKDM1A
SCHEMBL9865137 0.87 NAMPT (0.68) NAMPTHDAC1HDAC2HDAC3NR1H4
SCHEMBL9866050 0.86 GAA (0.54) LMNAKDM1AMAOAKDM1BRCOR1
SCHEMBL9865717 0.83 KDM1A (0.48) PAX8NR1H4LMNAKDM1AMAOA
SCHEMBL9865134 0.83 HTT (0.53) PAX8ALDH1A1HPGDHTT
SCHEMBL9335791 0.82 HTT (0.49) HDAC1HDAC2HDAC3PAX8HTT
SCHEMBL9335708 0.82 NR1H4 (0.49) PAX8NR1H4LMNAKDM1AMAOA
SCHEMBL9867342 0.82 NAMPT (0.59) NAMPTHDAC1HDAC2HDAC3NR1H4
SCHEMBL9867129 0.82 HDAC6 (0.49) HDAC1HDAC2HDAC3PAX8HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5039805-A Novel benzoic and phenylacetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1991-08-13 US disclosed
EP-0372486-A2 Benzoic-acid phenylacetic-acid derivatives, their preparation and their use as medicines F. HOFFMANN-LA ROCHE AG (CH) 1990-06-13 EP disclosed