SCHEMBL9867089

SCHEMBL9867089

Cc1coc2c(C(=O)c3ccccc3)cc(C(C)(C)C)c(O)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.41
HSD17B10 Q99714 3/20 0.41
KDM4E B2RXH2 3/20 0.41
LMNA P02545 2/20 0.41
PKM P14618 2/20 0.41
HPGD P15428 2/20 0.41
USP2 O75604 2/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 2/20 0.41
ALOX15 P16050 2/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41
XBP1 P17861 1/20 0.41
HTT P42858 1/20 0.41
TNFRSF1A P19438 1/20 0.38
ALOX5 P09917 2/20 0.37
PTGS1 P23219 2/20 0.37
PTGS2 P35354 2/20 0.37
BCL2 P10415 1/20 0.37
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867836 0.88 SIRT1 (0.46) MAPK1HSD17B10KDM4ELMNAPKM
SCHEMBL9866780 0.82 ALOX5 (0.55) HSD17B10KDM4ELMNAHPGDUSP2
SCHEMBL9867950 0.78 NPC1 (0.38) KDM4EHPGDPOLBTNFRSF1AALOX5
SCHEMBL9866482 0.76 LMNA (0.50) MAPK1HSD17B10KDM4ELMNAPKM
SCHEMBL9867508 0.75 NPC1 (0.45) HSD17B10KDM4EHPGDGAAMAPT
SCHEMBL9868331 0.75 CYP2C9 (0.44) HSD17B10KDM4ELMNAGAAMAPT
SCHEMBL10868061 0.73 TNFRSF1A (0.46) MAPK1HSD17B10KDM4ELMNAHPGD
SCHEMBL8420546 0.73 TNFRSF1A (0.48) MAPK1HSD17B10KDM4ELMNAHPGD
SCHEMBL4113584 0.72 GLRA3 (0.54) MAPK1HSD17B10KDM4ELMNAUSP2
SCHEMBL11211507 0.72 BCL2 (0.47) MAPK1HSD17B10KDM4ELMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006549-A Antiinflammatory agents MERCK & CO., INC. (US) 1991-04-09 US claimed
US-5006549-A Antiinflammatory agents MERCK & CO., INC. (US) 1991-04-09 US disclosed
EP-0399773-A1 Novel 7-aroyl-4-hydroxy-3-methyl benzolfurans as dual inhibitors of cyclooxygenase and 5-lipoxygenase MERCK & CO. INC. (US) 1990-11-28 EP disclosed