SCHEMBL9867950

SCHEMBL9867950

Cc1c(C(=O)O)oc2c(C(=O)c3ccccc3)cc(C(C)(C)C)c(O)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
MCL1 Q07820 3/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
TNFRSF1A P19438 1/20 0.36
GLRA3 O75311 1/20 0.36
GLRB P48167 1/20 0.36
ALOX5 P09917 3/20 0.36
PTGS1 P23219 2/20 0.36
PTGS2 P35354 2/20 0.36
BCL2 P10415 1/20 0.36
EDNRA P25101 1/20 0.35
AKR1C3 P42330 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868574 0.90 MCL1 (0.39) NPC1RAB9AL3MBTL1MEN1KMT2A
SCHEMBL9867508 0.87 NPC1 (0.45) NPC1RAB9AL3MBTL1ALDH1A1KDM4E
SCHEMBL9869017 0.84 ALOX5 (0.52) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL9868498 0.81 GLRA3 (0.49) L3MBTL1MEN1KMT2AALDH1A1KDM4E
SCHEMBL9867089 0.78 MAPK1 (0.41) RAB9AL3MBTL1MEN1KMT2AALDH1A1
SCHEMBL9867051 0.76 RAB9A (0.41) NPC1RAB9AL3MBTL1KMT2AALDH1A1
SCHEMBL4113584 0.76 GLRA3 (0.54) MEN1KMT2AALDH1A1KDM4EMCL1
SCHEMBL10868061 0.74 TNFRSF1A (0.46) MEN1KMT2AALDH1A1KDM4EHPGD
SCHEMBL9866663 0.71 ALOX5 (0.47) NPC1RAB9AL3MBTL1MEN1KMT2A
SCHEMBL9869198 0.71 EDNRA (0.47) NPC1RAB9AL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006549-A Antiinflammatory agents MERCK & CO., INC. (US) 1991-04-09 US disclosed
EP-0399773-A1 Novel 7-aroyl-4-hydroxy-3-methyl benzolfurans as dual inhibitors of cyclooxygenase and 5-lipoxygenase MERCK & CO. INC. (US) 1990-11-28 EP disclosed