SCHEMBL9868331

SCHEMBL9868331

Cc1coc2c(C(C)(C)C)cc(C(C)(C)C)c(O)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.44
CYP2C19 P33261 4/20 0.44
CYP1A2 P05177 2/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
CA2 P00918 3/20 0.44
ALDH1A1 P00352 3/20 0.44
POLB P06746 1/20 0.44
TYR P14679 1/20 0.44
CA1 P00915 2/20 0.41
GLRA3 O75311 1/20 0.39
GLRB P48167 1/20 0.39
HSPA5 P11021 2/20 0.39
MAPT P10636 2/20 0.36
ALOX15 P16050 2/20 0.36
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
HPN P05981 1/20 0.36
SIRT5 Q9NXA8 1/20 0.36
HIF1A Q16665 3/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2269577 0.75 ALDH1A1 (0.37) CYP2C9CYP2C19CYP1A2SMN1; SMN2CA2
SCHEMBL9866780 0.75 ALOX5 (0.55) ALDH1A1MAPTALOX15HSD17B10KDM4E
SCHEMBL9867089 0.75 MAPK1 (0.41) SMN1; SMN2ALDH1A1POLBMAPTALOX15
SCHEMBL9867836 0.73 SIRT1 (0.46) CYP2C9CYP2C19CYP1A2SMN1; SMN2ALDH1A1
SCHEMBL2268415 0.71 GABRA1 (0.44) CYP2C9CYP2C19CYP1A2SMN1; SMN2CA2
SCHEMBL16649211 0.71 ALDH1A1 (0.37) CYP2C9CYP2C19CYP1A2SMN1; SMN2CA2
SCHEMBL9244593 0.67 SMN1; SMN2 (0.64) CYP2C9CYP2C19CYP1A2SMN1; SMN2CA2
SCHEMBL20657093 0.66 CA2 (0.65) CYP2C9CYP2C19CYP1A2SMN1; SMN2CA2
SCHEMBL9868498 0.66 GLRA3 (0.49) CYP2C9CYP2C19CYP1A2SMN1; SMN2CA2
SCHEMBL29462687 0.64 CA2 (0.62) CYP2C9CYP2C19CYP1A2SMN1; SMN2CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006549-A Antiinflammatory agents MERCK & CO., INC. (US) 1991-04-09 US disclosed
EP-0399773-A1 Novel 7-aroyl-4-hydroxy-3-methyl benzolfurans as dual inhibitors of cyclooxygenase and 5-lipoxygenase MERCK & CO. INC. (US) 1990-11-28 EP disclosed