SCHEMBL9869490

SCHEMBL9869490

OC(=S)c1cccnc1Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
POLB P06746 1/20 0.42
ALDH1A1 P00352 3/20 0.41
PAX8 Q06710 1/20 0.41
CYP2C9 P11712 1/20 0.41
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
ALOX12 P18054 1/20 0.39
MET P08581 1/20 0.38
CALM1 P0DP23 1/20 0.38
LMNA P02545 1/20 0.38
NSD2 O96028 1/20 0.37
FABP1 P07148 1/20 0.37
FABP6 P51161 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
L3MBTL1 Q9Y468 4/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
CASP3 P42574 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869489 0.82 L3MBTL1 (0.44) KDM4EPOLBALDH1A1RAB9ASMN1; SMN2
SCHEMBL258223 0.82 ALDH1A1 (0.55) KDM4EPOLBALDH1A1CYP2C9RAB9A
SCHEMBL158842 0.82 POLB (0.49) KDM4EPOLBALDH1A1PAX8CYP2C9
SCHEMBL2306128 0.79 SYK (0.48) KDM4EPOLBALDH1A1CYP2C9RAB9A
SCHEMBL9869486 0.79 POLB (0.47) KDM4EPOLBALDH1A1PAX8CYP2C9
SCHEMBL5739085 0.78 KDM4E (0.38) KDM4EPOLBALDH1A1RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL11508163 0.77 SYK (0.46) KDM4EPOLBALDH1A1CYP2C9RAB9A
SCHEMBL4489937 0.77 P2RX7 (0.55) KDM4EPOLBALDH1A1CYP2C9RAB9A
SCHEMBL4500023 0.76 L3MBTL1 (0.60) KDM4EPOLBALDH1A1CYP2C9RAB9A
SCHEMBL9869479 0.76 L3MBTL1 (0.47) KDM4EPOLBALDH1A1CYP2C9RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006532-A Enzyme inhibitor; antiinflammatory agents MERCK & CO. INC., INC. (US) 1991-04-09 US disclosed
US-4904672-A Derivatives of 3-hydroxyazabenzo[b]thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1990-02-27 US disclosed
US-4767766-A Derivatives of 3-hydroxyazabenzo(B)thiophene useful as 5-lipoxygenase inhibitors MERCK & CO., INC. (US) 1988-08-30 US disclosed