SCHEMBL9870929

SCHEMBL9870929

CCN1C(=S)NC(C)=C(C(=O)O)C1c1ccccc1N(C)C

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CACNA1F O60840 8/20 0.40
CACNA1D Q01668 8/20 0.40
CACNA1S Q13698 8/20 0.40
CACNA1C Q13936 8/20 0.40
ALDH1A1 P00352 4/20 0.40
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
GUSB P08236 1/20 0.35
DHFR P00374 1/20 0.33
CACNA1G O43497 1/20 0.33
KIF11 P52732 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871923 0.81 ALDH1A1 (0.54) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL9870085 0.73 GUSB (0.44) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL9870764 0.73 POLB (0.45) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL10913257 0.73 CACNA1F (0.51) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL9871999 0.71 ALDH1A1 (0.47) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL10358732 0.71 CACNA1D (0.58) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL9869503 0.71 CACNA1F (0.44) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL10359264 0.70 CACNA1C (0.50) CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9870739 0.70 ALDH1A1 (0.36) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1
SCHEMBL9869835 0.69 CACNA1F (0.68) CACNA1FCACNA1DCACNA1SCACNA1CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5071849-A Antiinflammatory, antianginal agent EGIS GYOGYSZERGYAR (HU) 1991-12-10 US disclosed