SCHEMBL9872968

SCHEMBL9872968

CN(C)Cc1cccc(CCCCN)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.52
NOS1 P29475 2/20 0.46
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
TAAR1 Q96RJ0 3/20 0.43
HRH1 P35367 2/20 0.42
SIGMAR1 Q99720 1/20 0.42
NOS3 P29474 1/20 0.40
GRIN2D O15399 2/20 0.40
GRIN3B O60391 2/20 0.40
GRIN1 Q05586 2/20 0.40
GRIN2A Q12879 2/20 0.40
GRIN2B Q13224 2/20 0.40
GRIN2C Q14957 2/20 0.40
GRIN3A Q8TCU5 2/20 0.40
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4449176 0.87 TAAR1 (0.57) NOS1ALDH1A1TSHRTAAR1HTR7
SCHEMBL30957025 0.82 MAOA (0.67) MAOANOS1TAAR1HRH1
SCHEMBL10988696 0.82 HTR7 (0.41) NOS1ALDH1A1TSHRTAAR1NOS3
Hydrochloric Acid SCHEMBL28919564 0.81 LPL (0.53) ALDH1A1TSHRSIGMAR1GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL8076952 0.81 LPL (0.53) ALDH1A1TSHRSIGMAR1GRIN2DGRIN3B
SCHEMBL989636 0.80 ALDH1A1 (0.67) NOS1ALDH1A1TSHRTAAR1GRIN2D
SCHEMBL9872121 0.80 SLC6A2 (0.48) NOS1ALDH1A1TSHRTAAR1GRIN2D
SCHEMBL12075404 0.79 MAOA (0.57) MAOATAAR1HRH1
SCHEMBL2464280 0.79 ALDH1A1 (0.54) NOS1ALDH1A1TSHRTAAR1NOS3
SCHEMBL10750679 0.78 NOS1 (0.50) NOS1ALDH1A1TSHRGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021429-A Histamine h2-antagonists; antisecretory-antiallergen agent; skin disorders and peptic ulcers ALLEN & HANSBURYS LIMITED (GB) 1991-06-04 US disclosed
US-4496567-A HSITAMINE H2 ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-01-29 US disclosed
EP-0013071-B1 PYRIMIDINONE DERIVATIVES, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-11-16 EP disclosed
EP-0013071-A1 Pyrimidinone derivatives, processes for preparing them and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-07-09 EP disclosed
WO-1980000966-A1 NEW HISTAMINE H2-ANTAGONISTS SMITH KLINE FRENCH LAB (GB) 1980-05-15 WO disclosed