SCHEMBL9873952

SCHEMBL9873952

CC(=O)c1c(NC(=O)c2ccc([N+](=O)[O-])cc2)cccc1C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.54
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
RXFP1 Q9HBX9 1/20 0.53
RORC P51449 1/20 0.50
KDR P35968 1/20 0.50
DUSP3 P51452 1/20 0.50
PTPN5 P54829 1/20 0.50
CASP6 P55212 1/20 0.50
PTPN11 Q06124 1/20 0.50
PLK1 P53350 1/20 0.49
PLK3 Q9H4B4 1/20 0.49
PARP1 P09874 1/20 0.48
HTT P42858 3/20 0.47
GAA P10253 2/20 0.47
LMNA P02545 2/20 0.47
CASP3 P42574 1/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
POLB P06746 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7373448 0.85 RORC (0.66) NPC1ALDH1A1MAPTRXFP1RORC
SCHEMBL9874486 0.84 MAPT (0.56) NPC1ALDH1A1MAPTRXFP1PLK1
SCHEMBL9875019 0.84 MEN1 (0.56) NPC1ALDH1A1MAPTRXFP1PLK1
SCHEMBL9872839 0.83 RAB9A (0.59) NPC1MAPTRXFP1KDRPLK1
SCHEMBL9874407 0.81 F10 (0.59) NPC1ALDH1A1MAPTRXFP1PLK1
SCHEMBL22734230 0.77 ALDH1A1 (0.65) NPC1ALDH1A1MAPTRXFP1RORC
SCHEMBL9872671 0.77 SMN1; SMN2 (0.49) MAPTPLK1PLK3GAALMNA
SCHEMBL9875470 0.76 ALDH1A1 (0.48) ALDH1A1MAPTKDRPLK1PLK3
SCHEMBL7372951 0.76 KMT2A (0.69) NPC1ALDH1A1MAPTRXFP1KDR
SCHEMBL26416850 0.76 ALDH1A1 (0.67) NPC1ALDH1A1MAPTRXFP1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017576-A Antianxiolytic, hypnotic, anticonvulsant, antiepileptic RHONE-POULENC SANTE (FR) 1991-05-21 US disclosed