SCHEMBL9874730

SCHEMBL9874730

CC(=O)c1c(NC(=O)C(C)(C)C)cccc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 1/20 0.46
POLB P06746 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 2/20 0.46
PDK1 Q15118 6/20 0.44
PDK2 Q15119 6/20 0.44
PDK3 Q15120 6/20 0.44
PDK4 Q16654 6/20 0.44
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PLK1 P53350 1/20 0.41
PLK3 Q9H4B4 1/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ATM Q13315 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4453238 0.88 PLK1 (0.52) CETPPOLBCYP1A2CYP2C9PDK1
SCHEMBL26628119 0.82 CETP (0.57) CETPPOLBCYP1A2CYP2C9KDM4E
SCHEMBL9457765 0.81 TAS2R14 (0.55) CETPPOLBCYP1A2CYP2C9PDK1
SCHEMBL30977681 0.81 TAS2R14 (0.55) CETPPOLBCYP1A2CYP2C9PDK1
SCHEMBL1995318 0.78 THRB (0.48) KDM4EMEN1KMT2ALMNAGAA
SCHEMBL9874486 0.77 MAPT (0.56) MEN1KMT2APLK1PLK3LMNA
SCHEMBL9875019 0.77 MEN1 (0.56) CYP1A2KDM4EMEN1KMT2APLK1
SCHEMBL9873262 0.77 CETP (0.44) CETPPOLBCYP1A2CYP2C9PDK1
SCHEMBL9872839 0.76 RAB9A (0.59) CYP1A2MEN1KMT2APLK1PLK3
SCHEMBL9872356 0.76 SMN1; SMN2 (0.52) KDM4EMEN1KMT2ALMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017576-A Antianxiolytic, hypnotic, anticonvulsant, antiepileptic RHONE-POULENC SANTE (FR) 1991-05-21 US disclosed