SCHEMBL9874835

SCHEMBL9874835

O=C1CC(c2cccc(F)c2)=Nc2cccc(C(F)(F)F)c21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
CYP3A4 P08684 4/20 0.40
GRM2 Q14416 2/20 0.40
GRM3 Q14832 1/20 0.40
CYP11B2 P19099 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9872637 0.87 MAPT (0.40) TP53MAPTTHRBPDE3BPDE3A
SCHEMBL9872713 0.85 CYP3A4 (0.41) CYP3A4GRM2GRM3
SCHEMBL9873453 0.82 P2RX7 (0.35) TP53MAPTTHRBSMN1; SMN2PDE3B
SCHEMBL9872038 0.81 NOTUM (0.36) TP53MAPTSMN1; SMN2PDE3BPDE3A
SCHEMBL9872061 0.81 RAB9A (0.45) MAPTSMN1; SMN2CYP3A4GRM2GRM3
SCHEMBL9874871 0.78 PDE3B (0.37) PDE3BPDE3A
SCHEMBL9875005 0.78 MAPT (0.42) TP53MAPTTHRBSMN1; SMN2CYP11B2
SCHEMBL340807 0.77 MAPT (0.51) TP53MAPTTHRBSMN1; SMN2
SCHEMBL9872580 0.77 MAPT (0.43) MAPTCYP3A4
SCHEMBL31490607 0.74 TP53 (0.47) TP53MAPTTHRBSMN1; SMN2PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017576-A Antianxiolytic, hypnotic, anticonvulsant, antiepileptic RHONE-POULENC SANTE (FR) 1991-05-21 US disclosed