SCHEMBL9901491

SCHEMBL9901491

Cc1onc2cccc(Oc3ccc(NC(=O)C(C)(C)N(C(=O)O)C(C)(C)C)cc3)c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.42
RAF1 P04049 4/20 0.37
MAPK14 Q16539 2/20 0.37
MAPK13 O15264 1/20 0.37
MAPK12 P53778 1/20 0.37
MAPK11 Q15759 1/20 0.37
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
TP53 P04637 1/20 0.36
BRAF P15056 1/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 2/20 0.35
POLB P06746 1/20 0.35
CRHBP P24387 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15303017 0.85 PTGS2 (0.38) PTGS2RAF1MAPK14MAPK13MAPK12
SCHEMBL9905617 0.84 PTGS2 (0.43) PTGS2RAF1MAPK14MAPK13MAPK12
SCHEMBL13721386 0.79 GAA (0.56) PDK1PDK2PDK3PDK4MEN1
SCHEMBL13720494 0.75 GAA (0.51) PDK1PDK2PDK3PDK4MEN1
SCHEMBL18581856 0.72 MTNR1B (0.60) RAF1PDK1PDK2PDK3PDK4
SCHEMBL9900752 0.69 ALDH1A1 (0.41) MEN1KMT2AALDH1A1GAAPOLB
SCHEMBL9924093 0.68 KIT (0.45) PTGS2RAF1MAPK14MAPK13MAPK12
SCHEMBL29438018 0.68 KIT (0.45) PTGS2RAF1MAPK14MAPK13MAPK12
SCHEMBL13721575 0.68 PKM (0.40) MEN1KMT2AALDH1A1GAAPOLB
SCHEMBL15303500 0.66 MET (0.38) PTGS2RAF1MAPK14MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649066-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS Autifony Therapeutics Limited (GB) 2013-10-16 EP disclosed
WO-2012076877-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS AUTIFONY THERAPEUTICS LIMITED (GB) 2012-06-14 WO disclosed