Edetic Acid

Edetic Acid

SCHEMBL991956

O.O=C([O-])CN(CCN(CC(=O)[O-])CC(=O)[O-])CC(=O)[O-].[Na+].[Na+].[Na+].[Na+]

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Edetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE known ✓ P12821 1/20 0.48
CHRM2 known ✓ P08172 1/20 0.46
ADRA2A known ✓ P08913 1/20 0.46
SLC6A2 known ✓ P23975 1/20 0.46
SLC6A4 known ✓ P31645 1/20 0.46
ADRA1A known ✓ P35348 1/20 0.46
DRD3 known ✓ P35462 1/20 0.46
SLC6A3 known ✓ Q01959 1/20 0.46
HDAC3 known ✓ O15379 1/20 0.33
HDAC1 known ✓ Q13547 1/20 0.33
HDAC2 known ✓ Q92769 1/20 0.33
HDAC8 known ✓ Q9BY41 1/20 0.33
KDM4E B2RXH2 2/20 0.73
ALOX15 P16050 2/20 0.73
MAPT P10636 1/20 0.73
SMN1; SMN2 Q16637 1/20 0.73
TDP1 Q9NUW8 2/20 0.48
EYA2 O00167 1/20 0.48
APP P05067 1/20 0.48
BLM P54132 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Edetic Acid SCHEMBL1714086 1.00 KDM4E (0.73) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL10607814 1.00 KDM4E (0.73) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL8374505 1.00 KDM4E (0.73) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL978169 1.00 KDM4E (0.73) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL7071979 1.00 KDM4E (0.73) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL506851 1.00 KDM4E (0.73) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL8470881 1.00 KDM4E (0.73) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL5273812 0.97 KDM4E (0.70) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL3394139 0.97 KDM4E (0.70) KDM4EALOX15MAPTSMN1; SMN2TDP1
Edetic Acid SCHEMBL17747958 0.97 KDM4E (0.70) KDM4EALOX15MAPTSMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 316 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118948757-A Sodium hyaluronate eye drops and preparation method thereof 博济医药科技股份有限公司 2024-11-15 CN claimed
CN-111295202-B External preparation for treating onychomycosis 科研制药株式会社 2022-07-08 CN claimed
WO-2021112240-A1 RHINENCHYSIS COMPOSITION CONTAINING OLOPATADINE 東興薬品工業株式会社 2021-06-10 WO claimed
WO-2021112242-A1 PHARMACEUTICAL COMPOSITION COMPRISING STEROID COMPOUND AND OLOPATADINE 東興薬品工業株式会社 2021-06-10 WO claimed
CN-112566635-A Granular composition and process for producing the same 日本脏器制药株式会社 2021-03-26 CN claimed
CN-111836627-A Composition for suppressing pollen cracking 参天制药株式会社 2020-10-27 CN claimed
CN-111712238-A Eye drops containing 2-amino-3- (4-bromobenzoyl) phenylacetic acid or its salt 参天制药株式会社 2020-09-25 CN claimed
CN-111295202-A External preparation for treating onychomycosis 科研制药株式会社 2020-06-16 CN claimed
WO-2020032159-A1 PARTICULATE COMPOSITION AND PRODUCTION METHOD THEREFOR 日本臓器製薬株式会社 2020-02-13 WO claimed
WO-2019176947-A1 POLLEN BURSTING-INHIBITING COMPOSITION 参天製薬株式会社 2019-09-19 WO claimed
WO-2012169849-A2 EYE-DROP COMPOSITION FOR PREVENTING OR TREATING OCULAR DISEASES HUONS CO., LTD. (KR) 2012-12-13 WO claimed
US-5449658-A Biocidal compositions comprising polyhexamethylene biguanide and EDTA, and methods for treating commercial and recreational water ZENECA, INC. (US) 1995-09-12 US claimed
WO-1995015683-A1 BIOCIDAL COMPOSITIONS AND METHODS FOR TREATING COMMERCIAL AND RECREATIONAL WATER ZENECA, INC. (US) 1995-06-15 WO claimed
US-20260116959-A1 PHARMACEUTICAL COMPOSITION COMPRISING ANTI-PD-L1 ANTIBODY USED IN COMBINATION WITH ANTI-VEGF ANTIBODY AND PACLITAXEL (as amended) CHUGAI PHARMACEUTICAL CO LTD (JP) 2026-04-30 US disclosed
US-20260098160-A1 WATER RESISTANCE FOR ORGANIC FACADES ROHM & HAAS (US) 2026-04-09 US disclosed
US-20260008775-A1 AZOLE MODULATORS OF CHOLESTEROL BIOSYNTHESIS AND THEIR USE FOR PROMOTING REMYELINATION CONVELO THERAPEUTICS, INC. 2026-01-08 US disclosed
EP-0702662-A1 METHOD FOR TREATING WATER USING AN ORGANIC SANITIZER AND A PERSULFATE FMC CORPORATION (US) 1996-03-27 EP disclosed
US-5501802-A SWIMMING POOL FMC CORPORATION (US) 1996-03-26 US disclosed
WO-1995015683-A1 BIOCIDAL COMPOSITIONS AND METHODS FOR TREATING COMMERCIAL AND RECREATIONAL WATER ZENECA, INC. (US) 1995-06-15 WO disclosed
WO-1994024054-A1 METHOD FOR TREATING WATER USING AN ORGANIC SANITIZER AND A PERSULFATE FMC CORPORATION (US) 1994-10-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260098160-A1 WATER RESISTANCE FOR ORGANIC FACADES ERG, LATS2, FTO ACE 3061/4885CHRM2 2644/4885ADRA2A 1814/4885
US-20260116959-A1 PHARMACEUTICAL COMPOSITION COMPRISING ANTI-PD-L1 ANTIBODY USED IN COMBINATION WITH ANTI-VEGF ANTIBODY AND PACLITAXEL (as amended) PDCD1LG2, CD274, PDCD1 ACE 3251/4885CHRM2 2403/4885ADRA2A 1008/4885
US-20260008775-A1 AZOLE MODULATORS OF CHOLESTEROL BIOSYNTHESIS AND THEIR USE FOR PROMOTING REMYELINATION MAG, NR1H3, NR1H2 ACE 4489/4885CHRM2 278/4885ADRA2A 2808/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.