SCHEMBL9953497

SCHEMBL9953497

Cc1cccc(C)c1-n1c(N)nc2ccc(I)cc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.43
HCAR1 Q9BXC0 5/20 0.41
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PI4KA P42356 1/20 0.38
PIK3CG P48736 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954830 0.92 HCAR1 (0.43) PDE4DHCAR1CA12CA1CA2
SCHEMBL9954001 0.86 PDE4D (0.56) PDE4DHCAR1CA12CA1CA2
SCHEMBL9954005 0.84 HCAR1 (0.40) PDE4DHCAR1CA12CA1CA2
SCHEMBL9954505 0.84 PDE7A (0.45) PDE4DHCAR1PI4KA
SCHEMBL9953324 0.81 HCAR1 (0.50) HCAR1CA12CA1CA2CA9
SCHEMBL9953800 0.80 POLB (0.41) PDE4DHCAR1CA12CA1CA2
SCHEMBL9954358 0.80 ALDH1A1 (0.53) PDE4DHCAR1CA12CA1CA2
SCHEMBL9954224 0.79 CDK9 (0.38) PDE4DHCAR1CA12CA1CA2
SCHEMBL9953432 0.78 HCAR1 (0.55) PDE4DHCAR1KDM4EALDH1A1LMNA
SCHEMBL9953795 0.78 SMN1; SMN2 (0.55) KDM4EALDH1A1LMNAPI4KAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed