SCHEMBL9954830

SCHEMBL9954830

Cc1cccc(Cl)c1-n1c(N)nc2ccc(I)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 6/20 0.43
EPHB4 P54760 1/20 0.41
PDE4D Q08499 1/20 0.39
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
CDK9 P50750 1/20 0.37
DYRK1A Q13627 1/20 0.37
DYRK2 Q92630 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
PI4KA P42356 1/20 0.37
PIK3CG P48736 1/20 0.37
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
IDO2 Q6ZQW0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953497 0.92 PDE4D (0.43) HCAR1PDE4DCA12CA1CA2
SCHEMBL9954224 0.88 CDK9 (0.38) HCAR1EPHB4PDE4DCA12CA1
SCHEMBL9954005 0.82 HCAR1 (0.40) HCAR1PDE4DCA12CA1CA2
SCHEMBL9954001 0.81 PDE4D (0.56) HCAR1PDE4DCA12CA1CA2
SCHEMBL9954747 0.81 HCAR1 (0.53) HCAR1
SCHEMBL9954505 0.79 PDE7A (0.45) HCAR1PDE4DDYRK1API4KATDO2
SCHEMBL9953324 0.76 HCAR1 (0.50) HCAR1CA12CA1CA2CA9
SCHEMBL9953800 0.75 POLB (0.41) HCAR1PDE4DCA12CA1CA2
SCHEMBL9954358 0.75 ALDH1A1 (0.53) HCAR1PDE4DCA12CA1CA2
SCHEMBL9953432 0.73 HCAR1 (0.55) HCAR1PDE4DTDO2IDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed