SCHEMBL9954358

SCHEMBL9954358

Cc1ccc(-n2c(N)nc3ccc(I)cc3c2=O)c(C)c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.53
KDM4E B2RXH2 1/20 0.52
MAPT P10636 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HPD P32754 2/20 0.45
POLB P06746 1/20 0.41
PDE4D Q08499 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDO2 P48775 1/20 0.41
IDO2 Q6ZQW0 1/20 0.41
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
HCAR1 Q9BXC0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953564 0.88 TDO2 (0.48) ALDH1A1HPDPOLBPDE4DTDO2
SCHEMBL9953739 0.88 HPD (0.47) ALDH1A1KDM4EMAPTSMN1; SMN2HPD
SCHEMBL9954001 0.86 PDE4D (0.56) ALDH1A1KDM4EMAPTSMN1; SMN2HPD
SCHEMBL9954234 0.85 ALDH1A1 (0.53) ALDH1A1KDM4EMAPTSMN1; SMN2HPD
SCHEMBL9953800 0.81 POLB (0.41) POLBPDE4DCA12CA1CA2
SCHEMBL9953497 0.80 PDE4D (0.43) ALDH1A1KDM4EPDE4DCA12CA1
SCHEMBL9952904 0.78 GLA (0.51) MAPTPOLBTDO2IDO2HCAR1
SCHEMBL9954671 0.77 HCAR1 (0.52) HPDPDE4DTDO2IDO2HCAR1
SCHEMBL9954747 0.76 HCAR1 (0.53) ALDH1A1KDM4ESMN1; SMN2HPDPOLB
SCHEMBL9953432 0.76 HCAR1 (0.55) ALDH1A1KDM4EMAPTPOLBPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed