SCHEMBL9956413

SCHEMBL9956413

Cc1nc(C=O)c(-c2cccc(F)c2)o1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.39
PTGS2 P35354 2/20 0.39
TRPM8 Q7Z2W7 2/20 0.39
PDE4B Q07343 2/20 0.38
PTGS1 P23219 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
MGAM O43451 1/20 0.37
GAA P10253 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
MAOB P27338 1/20 0.36
NR4A1 P22736 1/20 0.36
NR4A2 P43354 1/20 0.36
NR4A3 Q92570 1/20 0.36
FPR2 P25090 1/20 0.36
SLC9A1 P19634 1/20 0.36
IDO1 P14902 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9955506 0.85 RAB9A (0.41) NOTUMGAAMAOBNR4A2IDO1
SCHEMBL9955896 0.82 NOTUM (0.39) NOTUMPDE4BMGAMGAASI
SCHEMBL5543913 0.80 TRPM8 (0.43) NOTUMPTGS2TRPM8PTGS1MGAM
SCHEMBL5543906 0.77 TRPM8 (0.41) NOTUMPTGS2TRPM8PTGS1MGAM
SCHEMBL1167044 0.75 PIN1 (0.50) TRPM8PDE4BNR4A1NR4A2NR4A3
SCHEMBL10263245 0.75 TRPM8 (0.42) NOTUMPTGS2TRPM8PTGS1MGAM
SCHEMBL7624713 0.75 PTGS2 (0.59) PTGS2TRPM8PTGS1
SCHEMBL10263340 0.73 L3MBTL1 (0.45) TRPM8MGAMGAASIMGAM2
SCHEMBL31194857 0.73 MAPK13 (0.60) PTGS2PTGS1NR4A2
SCHEMBL9956374 0.73 NOTUM (0.44) NOTUMNR4A1NR4A2NR4A3IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed