SCHEMBL9963456

SCHEMBL9963456

CC(C)NC(=O)C(C)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.41
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA12 O43570 1/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
CA9 Q16790 1/20 0.37
TSHR P16473 1/20 0.37
ALDH1A1 P00352 3/20 0.34
GAA P10253 1/20 0.34
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
MLYCD O95822 1/20 0.31
CA7 P43166 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16015868 1.00 DPP4 (0.41) DPP4CA1CA2CA12MMP1
SCHEMBL9963462 0.82 DPP4 (0.39) DPP4CA1CA2ALDH1A1POLB
SCHEMBL19507003 0.80 CA12 (0.34) DPP4CA1CA2CA12MMP1
SCHEMBL22080181 0.80 CA12 (0.34) DPP4CA1CA2CA12MMP1
SCHEMBL12212142 0.78 ALDH1A1 (0.35) CA1CA2CA12MMP1MMP2
SCHEMBL13691202 0.78 MME (0.46) DPP4LMNA
SCHEMBL19845930 0.77 MMP1 (0.36) DPP4CA1CA2CA12MMP1
SCHEMBL20907635 0.77 MLYCD (0.38) CA1CA2CA12MMP1MMP2
SCHEMBL21149312 0.77 MLYCD (0.38) CA1CA2CA12MMP1MMP2
SCHEMBL12884385 0.77 CA1 (0.41) DPP4CA1CA2CA12MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11655239-B2 Fused ring pyrimidine amino compound and preparation method, pharmaceutical composition, and use thereof Shanghai Institute of Material Medica, Chinese Academy of Sciences (CN) 2023-05-23 US disclosed
US-20170355797-A1 MOLECULARLY IMPRINTED COPOLYMER COMPOUNDS AND METHODS OF PREPARATION AND USE THEREOF UNIVERSITY OF NEW HAMPSHIRE (US) 2017-12-14 US disclosed
US-8354403-B2 Pyrrolidine derived beta 3 adrenergic receptor agonists MERCK SHARP & DOHME CORP. (US) 2013-01-15 US disclosed
US-20120157432-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME, CORP. (US) 2012-06-21 US disclosed
US-20110028447-A1 INDAZOLE DERIVATIVES PFIZER INC. 2011-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120157432-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS ADRB3, ADRB1, ADRB2 DPP4 1841/4885CA1 4877/4885CA2 4152/4885
US-20110028447-A1 INDAZOLE DERIVATIVES CNR1, CNR2, GPR119 DPP4 3705/4885CA1 2678/4885CA2 1778/4885
US-11655239-B2 Fused ring pyrimidine amino compound and preparation method, pharmaceutical composition, and use thereof DDR2, DDR1, DOCK2 DPP4 1931/4885CA1 4883/4885CA2 4372/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.