SCHEMBL9970109

SCHEMBL9970109

Cc1cnc(C)c(C)c1CN

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
AOC3 Q16853 8/20 0.41
KDM4E B2RXH2 2/20 0.37
AOC1 P19801 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
LOX P28300 2/20 0.32
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
AGXT P21549 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12319209 0.79 NOS3 (0.38) KDM4ENOS3NOS1NOS2CCR1
SCHEMBL15142288 0.78 LMNA (0.42) LMNAAOC3AOC1NOS3NOS1
SCHEMBL9970101 0.78 LMNA (0.50) LMNAAOC3KDM4EAOC1LOX
SCHEMBL14682728 0.78 LMNA (0.65) LMNAAOC3KDM4EAOC1NOS3
SCHEMBL9970098 0.75 LMNA (0.71) LMNAAOC3KDM4ELOXALDH1A1
Ethylenediamine SCHEMBL6295958 0.74 CCR1 (0.38) LMNAKDM4ENOS3NOS1NOS2
SCHEMBL17229270 0.74 KDM5A (0.32) CCR1CCR5CCR8
SCHEMBL9970114 0.71 DPP4 (0.43) LMNAAOC3
SCHEMBL3671331 0.70 NOS3 (0.44) KDM4ENOS3NOS1NOS2CCR1
SCHEMBL22972190 0.70 AOC3 (0.48) LMNAAOC3AOC1LOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110003101-A A kind of Ah pa is for Buddhist nun's intermediate and preparation method thereof 苏州富士莱医药股份有限公司 2019-07-12 CN disclosed
US-20180153827-A1 COMPOSITIONS AND METHODS OF USE OF GAMMA-KETOALDEHYDE SCAVENGERS FOR TREATING, PREVENTING OR IMPROVING NONALCOHOLIC FATTY LIVER DISEASE (NAFLD), NASH, ALD OR CONDITIONS RELATED TO THE LIVER MTI BIOTECH, INC. 2018-06-07 US disclosed
US-20140256774-A1 METHODS FOR TREATING INFLAMMATION AND HYPERTENSION WITH GAMMA-KETOALDEHYDE SKAVENGERS VANDERBILT UNIVERSITY (US) 2014-09-11 US disclosed
US-8822542-B2 Isoketal scavengers and mitigation of disorders involving oxidative injury VANDERBILT UNIVERSITY (US) 2014-09-02 US disclosed
US-20120157501-A1 ISOKETAL SCAVENGERS AND MITIGATION OF DISORDERS INVOLVING OXIDATIVE INJURY VANDERBILT UNIVERSITY 2012-06-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140256774-A1 METHODS FOR TREATING INFLAMMATION AND HYPERTENSION WITH GAMMA-KETOALDEHYDE SKAVENGERS AKR1B1, NFKBIA, PTGS2 LMNA 1062/4885AOC3 706/4885KDM4E 607/4885
US-20120157501-A1 ISOKETAL SCAVENGERS AND MITIGATION OF DISORDERS INVOLVING OXIDATIVE INJURY PDXK, KYNU, FN3K LMNA 2014/4885AOC3 501/4885KDM4E 1534/4885
US-20180153827-A1 COMPOSITIONS AND METHODS OF USE OF GAMMA-KETOALDEHYDE SCAVENGERS FOR TREATING, PREVENTING OR IMPROVING NONALCOHOLIC FATTY LIVER DISEASE (NAFLD), NASH, ALD OR CONDITIONS RELATED TO THE LIVER CPT1A, AKR7A2, FABP1 LMNA 703/4885AOC3 480/4885KDM4E 692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.