SCHEMBL10014501

SCHEMBL10014501

c1ccc(-c2cccc(-n3c4ccccc4c4c5sc6ccccc6c5ccc43)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
ALOX5 P09917 1/20 0.36
MAPT P10636 4/20 0.35
RXFP1 Q9HBX9 1/20 0.35
TP53 P04637 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HTT P42858 2/20 0.33
HSD17B10 Q99714 1/20 0.33
FAAH O00519 1/20 0.33
HSP90AA1 P07900 1/20 0.33
PKM P14618 1/20 0.33
MGLL Q99685 1/20 0.33
GPR3 P46089 1/20 0.32
LIMK1 P53667 2/20 0.32
KMT2A Q03164 2/20 0.32
IL1R1 P14778 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16171123 0.98 ALOX5 (0.37) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL16171205 0.97 ALOX5 (0.37) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL24676263 0.96 KDM4E (0.39) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL19678247 0.95 ATM (0.38) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL16482212 0.95 ATM (0.38) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL24676276 0.95 ALOX5 (0.37) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL16283068 0.94 L3MBTL1 (0.40) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL19678252 0.94 TNKS (0.35) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL16482480 0.94 KDM4E (0.37) ATML3MBTL1KDM4ETNKSTNKS2
SCHEMBL24676345 0.94 KDM4E (0.39) ATML3MBTL1KDM4ETNKSTNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357150-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-11-09 US disclosed
US-20230357150-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO., LTD. (KR) 2023-11-09 US disclosed
US-20230363268-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-11-09 US disclosed
US-20230363268-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-11-09 US disclosed
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2023-09-28 US disclosed
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2023-09-28 US disclosed
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-09-21 US disclosed
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE SAMSUNG DISPLAY CO., LTD. (KR) 2023-09-21 US disclosed
US-20230225142-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2023-07-13 US disclosed
US-20230225142-A1 ORGANIC LIGHT-EMITTING DEVICE SAMSUNG ELECTRONICS CO LTD (KR) 2023-07-13 US disclosed
US-20150228909-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG SDI CO., LTD. (KR) 2015-08-13 US disclosed
WO-2015108301-A1 FUSED RING COMPOUND AND ORGANIC LIGHT EMITTING DEVICE COMPRISING SAME 삼성에스디아이 주식회사 2015-07-23 WO disclosed
WO-2015105316-A1 FUSED-RING COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME 삼성에스디아이 주식회사 2015-07-16 WO disclosed
EP-2894157-A1 Condensed cyclic compound and organic light-emitting device including the same Samsung Electronics Co., Ltd (KR) 2015-07-15 EP disclosed
US-20150053960-A1 COMPOUND CONTAINING A 5-MEMBERED HETEROCYCLE AND ORGANIC LIGHT-EMITTING DIODE USING SAME, AND TERMINAL FOR SAME DUK SAN NEOLUX CO., LTD. (KR) 2015-02-26 US disclosed
US-20150053960-A1 COMPOUND CONTAINING A 5-MEMBERED HETEROCYCLE AND ORGANIC LIGHT-EMITTING DIODE USING SAME, AND TERMINAL FOR SAME DUK SAN NEOLUX CO., LTD. (KR) 2015-02-26 US disclosed
US-8889271-B2 Compound containing a 5-membered heterocycle and organic light-emitting diode using same, and terminal for same DUKSAN HIGH METAL CO., LTD. (KR) 2014-11-18 US disclosed
US-8889271-B2 Compound containing a 5-membered heterocycle and organic light-emitting diode using same, and terminal for same DUKSAN HIGH METAL CO., LTD. (KR) 2014-11-18 US disclosed
US-20120080670-A1 COMPOUND CONTAINING A 5-MEMBERED HETEROCYCLE AND ORGANIC LIGHT-EMITTING DIODE USING SAME, AND TERMINAL FOR SAME SAMSUNG MOBILE DISPLAY CO., LTD. (KR) 2012-04-05 US disclosed
US-20120080670-A1 COMPOUND CONTAINING A 5-MEMBERED HETEROCYCLE AND ORGANIC LIGHT-EMITTING DIODE USING SAME, AND TERMINAL FOR SAME SAMSUNG MOBILE DISPLAY CO., LTD. (KR) 2012-04-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230225142-A1 ORGANIC LIGHT-EMITTING DEVICE EML4, ICMT, L1CAM ATM 3879/4885L3MBTL1 36/4885KDM4E 1380/4885
US-20150228909-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME CRY1, CCNE2, CRY2 ATM 1406/4885L3MBTL1 646/4885KDM4E 2145/4885
US-20230357150-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE AOX1, CRY1, CYP1A1 ATM 3294/4885L3MBTL1 1123/4885KDM4E 1958/4885
US-20230309390-A1 ORGANIC LIGHT-EMITTING DEVICE L1CAM, EML4, OR10J3 ATM 2243/4885L3MBTL1 23/4885KDM4E 2238/4885
US-20230363268-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE AOX1, CYP1A1, CRY1 ATM 3588/4885L3MBTL1 966/4885KDM4E 2677/4885
US-20230301179-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME, AND ELECTRONIC APPARATUS INCLUDING THE ORGANIC LIGHT-EMITTING DEVICE CRY1, AOX1, CYP1A1 ATM 3264/4885L3MBTL1 1020/4885KDM4E 2808/4885
US-20120080670-A1 COMPOUND CONTAINING A 5-MEMBERED HETEROCYCLE AND ORGANIC LIGHT-EMITTING DIODE USING SAME, AND TERMINAL FOR SAME NOTUM, OR10J3, PER2 ATM 3651/4885L3MBTL1 2162/4885KDM4E 1424/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.