SCHEMBL10069628

SCHEMBL10069628

CC(C)c1c(-c2cccs2)n(COCc2ccc(F)cc2)c(=O)n(O)c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.35
USP2 O75604 4/20 0.35
CYP3A4 P08684 4/20 0.35
CASP1 P29466 4/20 0.35
CASP7 P55210 4/20 0.35
CYP1A2 P05177 3/20 0.35
CYP2D6 P10635 3/20 0.35
HIF1A Q16665 3/20 0.35
HSD17B10 Q99714 3/20 0.35
TSHR P16473 2/20 0.35
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
KDM5B Q9UGL1 1/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 3/20 0.33
HBB P68871 2/20 0.33
GLA P06280 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
NPC1 O15118 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069604 0.91 ERCC5 (0.38) ALDH1A1USP2CYP3A4CASP1CASP7
SCHEMBL10069619 0.84 KDM5B (0.34) CYP3A4KDM5BTP53MAPTGNRHR
SCHEMBL10069611 0.84 L3MBTL1 (0.36) ALDH1A1USP2CYP3A4CYP1A2TSHR
SCHEMBL10069601 0.82 ALDH1A1 (0.36) ALDH1A1CYP3A4CASP1CASP7CYP1A2
SCHEMBL10069631 0.81 RGS4 (0.34) ALDH1A1KDM5BKMT2ASMN1; SMN2KDM4E
SCHEMBL10069627 0.80 ALDH1A1 (0.34) ALDH1A1HSD17B10MEN1KMT2ASMN1; SMN2
SCHEMBL10069596 0.80 MAPT (0.36) ALDH1A1USP2CYP3A4CASP1CASP7
SCHEMBL10069598 0.80 TP53 (0.33) TP53MAPT
SCHEMBL10069629 0.80 RGS4 (0.35) ALDH1A1TSHRLMNASMN1; SMN2KDM4E
SCHEMBL10069597 0.80 ANO1 (0.36) KDM5BLMNASMN1; SMN2MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed