SCHEMBL10071053

SCHEMBL10071053

CC(=O)N[C@@H](CC(=O)O)C(=O)NC(CCC(=O)O)C(=O)NC(C(=O)NC(CC(=O)O)C(=O)Nc1ccc([N+](=O)[O-])cc1)C(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDF Q9HBH1 1/20 0.43
CASP1 P29466 1/20 0.42
CASP3 P42574 1/20 0.42
CASP7 P55210 1/20 0.42
CASP9 P55211 1/20 0.42
MMP9 P14780 1/20 0.41
BACE1 P56817 9/20 0.41
BACE2 Q9Y5Z0 3/20 0.41
SSTR3 P32745 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
CTSD P07339 1/20 0.40
CTNNB1 P35222 1/20 0.40
MAPT P10636 2/20 0.39
LMNA P02545 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2028887 1.00 PDF (0.43) PDFCASP1CASP3CASP7CASP9
SCHEMBL18657234 1.00 PDF (0.43) PDFCASP1CASP3CASP7CASP9
SCHEMBL30910411 0.93 ENPEP (0.42) PDFCASP1CASP3CASP7CASP9
SCHEMBL22148813 0.92 SIRT5 (0.46) PDFSSTR3ALDH1A1
SCHEMBL22148827 0.92 SIRT5 (0.46) PDFSSTR3ALDH1A1
SCHEMBL3512725 0.91 BACE1 (0.46) PDFCASP1CASP3CASP7CASP9
SCHEMBL7885355 0.89 MMP9 (0.42) PDFCASP1MMP9BACE1BACE2
SCHEMBL29500567 0.89 PDF (0.45) PDFCASP1MMP9BACE1BACE2
SCHEMBL4594304 0.87 ENPEP (0.42) PDFBACE1SSTR3MEN1KMT2A
SCHEMBL7694593 0.83 CASP1 (0.56) CASP1CASP3CASP7BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120040995-A1 DESIGN, SYNTHESIS AND EVALUATION OF PROCASPASE ACTIVATING COMPOUNDS AS PERSONALIZED ANTI-CANCER DRUGS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120040995-A1 DESIGN, SYNTHESIS AND EVALUATION OF PROCASPASE ACTIVATING COMPOUNDS AS PERSONALIZED ANTI-CANCER DRUGS CASP3, CASP6, CASP14 PDF 144/4885CASP1 13/4885CASP3 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.