SCHEMBL1011540

SCHEMBL1011540

O=C(Nc1ccccn1)Oc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.59
NPC1 O15118 7/20 0.59
PKM P14618 3/20 0.59
GAA P10253 1/20 0.56
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
ADORA3 P0DMS8 1/20 0.56
PIM1 P11309 1/20 0.56
ADORA2A P29274 1/20 0.56
ADORA2B P29275 1/20 0.56
ADORA1 P30542 1/20 0.56
FLT3 P36888 1/20 0.56
PIM3 Q86V86 1/20 0.56
AURKB Q96GD4 1/20 0.56
ALDH1A1 P00352 2/20 0.54
F2 P00734 2/20 0.53
F12 P00748 1/20 0.53
KDM4E B2RXH2 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31286005 1.00 RAB9A (0.59) RAB9ANPC1PKMGAAMEN1
SCHEMBL16238273 0.87 NPC1 (0.60) RAB9ANPC1PKMGAAMEN1
SCHEMBL29874075 0.87 DHODH (0.55) RAB9ANPC1PKMGAAMEN1
SCHEMBL29018750 0.84 RAB9A (0.61) RAB9ANPC1PKMGAAMEN1
SCHEMBL15899827 0.84 RAB9A (0.54) RAB9ANPC1PKMGAAMEN1
SCHEMBL31414640 0.84 F2 (0.57) RAB9ANPC1PKMGAAMEN1
SCHEMBL27716616 0.83 GAA (0.55) RAB9ANPC1PKMGAAMEN1
SCHEMBL20448089 0.83 RAB9A (0.59) RAB9ANPC1PKMGAAMEN1
SCHEMBL2477935 0.82 NPC1 (0.57) RAB9ANPC1PKMMEN1KMT2A
SCHEMBL896911 0.82 GAA (0.60) GAAMEN1KMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 129 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12630562-B2 Piperidylurea compounds and methods of use thereof ARCUS BIOSCIENCES, INC. (US) 2026-05-19 US disclosed
US-20260042777-A1 PIPERIDYLUREA COMPOUNDS AND METHODS OF USE THEREOF ARCUS BIOSCIENCES, INC. (US) 2026-02-12 US disclosed
US-20250243161-A1 DELIVERY OF THERAPEUTIC ALKALOID COMPOUNDS SENSORIUM THERAPEUTICS, INC. 2025-07-31 US disclosed
US-12269800-B2 Delivery of therapeutic alkaloid compounds SENSORIUM THERAPEUTICS, INC. (US) 2025-04-08 US disclosed
US-20250051277-A1 DELIVERY OF THERAPEUTIC ALKALOID COMPOUNDS SENSORIUM THERAPEUTICS, INC. 2025-02-13 US disclosed
US-12110278-B2 Selective JAK2 pseudokinase ligands and methods of use YALE UNIVERSITY (US) 2024-10-08 US disclosed
US-20240246910-A1 DELIVERY OF THERAPEUTIC ALKALOID COMPOUNDS SENSORIUM THERAPEUTICS, INC. 2024-07-25 US disclosed
US-20240216355-A1 PHARMACEUTICAL COMPOSITIONS FOR USE IN THE PREVENTION AND TREATMENT OF A DISEASE OR DISORDER CAUSED BY OR ASSOCIATED WITH ONE OR MORE PREMATURE TERMINATION CODONS MONTE ROSA THERAPEUTICS AG (CH) 2024-07-04 US disclosed
US-11999694-B2 Delivery of therapeutic alkaloid compounds SENSORIUM THERAPEUTICS, INC. (US) 2024-06-04 US disclosed
EP-4313047-A1 PHARMACEUTICAL COMPOSITIONS FOR USE IN THE PREVENTION AND TREATMENT OF A DISEASE OR DISORDER CAUSED BY OR ASSOCIATED WITH ONE OR MORE PREMATURE TERMINATION CODONS Monte Rosa Therapeutics, Inc. (US) 2024-02-07 EP disclosed
US-4563452-A ANTIINFLAMMATORY, ANALGESIC PROVESAN S.A. (CH) 1986-01-07 US disclosed
EP-0078839-A4 HETEROCYCLIC AMIDINOUREAS. RORER INTERNAT OVERSEAS INC (US) 1984-07-25 EP disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed
EP-0099770-A1 Oxazinobenzothiazine-6,6-dioxide derivatives, their preparation and their use as medicament PROVESAN S.A. (CH) 1984-02-01 EP disclosed
US-4396621-A ANALGESICS, ANTIIMFLAMMATORY AGENTS CIBA-GEIGY CORPORATION (US) 1983-08-02 US disclosed
EP-0078839-A1 HETEROCYCLIC AMIDINOUREAS RORER INTERNATIONAL (OVERSEAS) INC. (US) 1983-05-18 EP disclosed
WO-1982004047-A1 HETEROCYCLIC AMIDINOUREAS RORER INT OVERSEAS (US) 1982-11-25 WO disclosed
US-4320138-A ANTIINFLAMMATORY AGENTS FOR ARTHRITIS, GOUT CIBA-GEIGY CORPORATION (US) 1982-03-16 US disclosed
US-4260779-A ANALGESICS, ANTIINFLAMMATORY, DIURETICS CIBA-GEIGY CORPORATION (US) 1981-04-07 US disclosed
US-3931202-A Pyridyl phenyl-carbamate rodenticides ROHM AND HAAS COMPANY (US) 1976-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12110278-B2 Selective JAK2 pseudokinase ligands and methods of use JAK2, JAK1, MCL1 RAB9A 4383/4885NPC1 4449/4885PKM 1321/4885
US-20250051277-A1 DELIVERY OF THERAPEUTIC ALKALOID COMPOUNDS PNMT, HNMT, NNMT RAB9A 571/4885NPC1 296/4885PKM 1751/4885
US-20240216355-A1 PHARMACEUTICAL COMPOSITIONS FOR USE IN THE PREVENTION AND TREATMENT OF A DISEASE OR DISORDER CAUSED BY OR ASSOCIATED WITH ONE OR MORE PREMATURE TERMINATION CODONS UPF1, NSUN2, RTF2 RAB9A 3771/4885NPC1 330/4885PKM 4089/4885
US-20250243161-A1 DELIVERY OF THERAPEUTIC ALKALOID COMPOUNDS PNMT, HNMT, NNMT RAB9A 571/4885NPC1 296/4885PKM 1751/4885
US-20240246910-A1 DELIVERY OF THERAPEUTIC ALKALOID COMPOUNDS PNMT, HNMT, NNMT RAB9A 571/4885NPC1 296/4885PKM 1751/4885
US-12630562-B2 Piperidylurea compounds and methods of use thereof CLIC1, HCCS, CNR1 RAB9A 767/4885NPC1 73/4885PKM 3271/4885
US-12269800-B2 Delivery of therapeutic alkaloid compounds PNMT, HNMT, NNMT RAB9A 571/4885NPC1 296/4885PKM 1751/4885
US-11999694-B2 Delivery of therapeutic alkaloid compounds PNMT, HNMT, NNMT RAB9A 571/4885NPC1 296/4885PKM 1751/4885
US-20260042777-A1 PIPERIDYLUREA COMPOUNDS AND METHODS OF USE THEREOF CBR1, CLIC1, RER1 RAB9A 485/4885NPC1 134/4885PKM 3398/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.