SCHEMBL10128

SCHEMBL10128

Clc1ccc(CBr)cc1Cl

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.58
PNMT P11086 2/20 0.54
TAAR1 Q96RJ0 1/20 0.54
SIGMAR1 Q99720 5/20 0.47
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
PYCR1 P32322 1/20 0.46
POLB P06746 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
IGF1R P08069 1/20 0.45
ALOX15 P16050 1/20 0.45
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
AHR P35869 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29413271 1.00 IDO1 (0.58) IDO1PNMTTAAR1SIGMAR1CYP4F2
SCHEMBL1964765 0.97 IDO1 (0.56) IDO1PNMTTAAR1SIGMAR1CYP4F2
SCHEMBL27276965 0.91 TP53 (0.61) IDO1PNMTTAAR1SIGMAR1CYP4F2
SCHEMBL4962307 0.82 SIGMAR1 (0.45) IDO1PNMTTAAR1SIGMAR1POLB
SCHEMBL30019331 0.80 PNMT (0.61) IDO1PNMTTAAR1SIGMAR1IGF1R
SCHEMBL507167 0.80 CYP4F2 (0.43) IDO1PNMTTAAR1SIGMAR1CYP4F2
SCHEMBL507688 0.80 CYP4F2 (0.40) IDO1PNMTTAAR1CYP4F2CYP4A11
SCHEMBL177296 0.80 PNMT (0.61) IDO1PNMTTAAR1SIGMAR1IGF1R
SCHEMBL30595364 0.80 CYP4F2 (0.40) IDO1PNMTTAAR1CYP4F2CYP4A11
SCHEMBL30488129 0.80 CYP4F2 (0.43) IDO1PNMTTAAR1SIGMAR1CYP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1370 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111004228-B GSK-3 beta/ChE double inhibitor and preparation method and application thereof 中国药科大学 2023-05-23 CN claimed
WO-2021047572-A1 GSK-3β/CHE DOUBLE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 中国药科大学 2021-03-18 WO claimed
CN-111004228-A GSK-3 β/ChE dual inhibitor and preparation method and application thereof 中国药科大学 2020-04-14 CN claimed
EP-4741397-A1 FUSED TRICYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF Shenzhen Zhongge Biological Technology Co., Ltd. (CN) 2026-05-13 EP disclosed
US-12570642-B2 GLP-IR modulating compounds GILEAD SCIENCES, INC. (US) 2026-03-10 US disclosed
EP-4691554-A2 GLP-1R MODULATING COMPOUNDS Gilead Sciences, Inc. (US) 2026-02-11 EP disclosed
EP-4271672-B1 CARBOXY-BENZIMIDAZOLE GLP-1R MODULATING COMPOUNDS GILEAD SCIENCES INC (US) 2025-12-03 EP disclosed
WO-2025243042-A1 COMPOUNDS FOR THE INHIBITION OF CYCLOPHILIN D THE UNIVERSITY OF LIVERPOOL (GB) 2025-11-27 WO disclosed
US-12473314-B2 Phospholipid compounds and uses thereof GILEAD SCIENCES, INC. (US) 2025-11-18 US disclosed
EP-4629980-A1 ANTIMICROBIAL COMPOUNDS SRI International (US) 2025-10-15 EP disclosed
US-20250205195-A1 BENZYLOXY-BENZYLAMINYL AMINO ACID DERIVATIVE FOR ADJUSTING TSLP/TSLPR SIGNAL TRANSMISSION AMTIXBIO CO., LTD. (KR) 2025-06-26 US disclosed
US-4279920-A 2,2-Dimethyl-3-(2-bromo-2-phenyl-vinyl)-cyclopropanecarboxylic acid 3-phenoxybenzyl esters and pesticidal use BAYER AKTIENGESELLSCHAFT (DE) 1981-07-21 US disclosed
EP-0001439-B1 1-N-SUBSTITUTED 1.4-DIHYDROPYRIDAZINE DERIVATIVES, METHOD FOR THEIR PREPARATION AND THEIR USE FOR PHARMACEUTICALS BAYER AG (DE) 1981-01-28 EP disclosed
US-RE30420-E DIURETIC, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DE) 1980-10-21 US disclosed
EP-0001439-A1 1-N-substituted 1.4-dihydropyridazine derivatives, method for their preparation and their use for pharmaceuticals BAYER AG (DE) 1979-04-18 EP disclosed
US-4112227-A DIURETIC, SALURETIC, ANTIHYPERTENSIVE, ANTITHROMBOTIC BAYER AKTIENGESELLSCHAFT (DE) 1978-09-05 US disclosed
US-4056533-A HYPOTENSIVE AGENTS, ANTICOAGULANTS, DIURETICS BAYER AKTIENGESELLSCHAFT (DT) 1977-11-01 US disclosed
US-4000294-A DIURESIS OR SALURESIS BAYER AKTIENGESELLSCHAFT (DT) 1976-12-28 US disclosed
US-3992404-A DIURETICS, SALURETICS, ANTIHYPERTENSIVE AGENTS, AND ANTITHROMBOTIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1976-11-16 US disclosed
US-3952008-A DIURETIC, SALURETIC, HYPOTENSIVE, ANTITHROMBOTIC BAYER AKTIENGESELLSCHAFT (DT) 1976-04-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12570642-B2 GLP-IR modulating compounds GLP1R, GIPR, GPR119 IDO1 2279/4885PNMT 3622/4885TAAR1 579/4885
US-12473314-B2 Phospholipid compounds and uses thereof PHOSPHO1, SGMS2, SGMS1 IDO1 3203/4885PNMT 665/4885TAAR1 4464/4885
US-20250205195-A1 BENZYLOXY-BENZYLAMINYL AMINO ACID DERIVATIVE FOR ADJUSTING TSLP/TSLPR SIGNAL TRANSMISSION TSLP, IL2RA, TRPC7 IDO1 781/4885PNMT 1638/4885TAAR1 345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.