SCHEMBL10539

SCHEMBL10539

CN(C)C(CC(Oc1ccc(C(F)(F)F)cc1)c1cccs1)OC(=O)C(=O)OC(CC(Oc1ccc(C(F)(F)F)cc1)c1cccs1)N(C)C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.52
SLC6A9 P48067 11/20 0.44
SLC6A4 P31645 2/20 0.41
HRH3 Q9Y5N1 2/20 0.41
TRPM8 Q7Z2W7 1/20 0.39
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
FFAR1 O14842 1/20 0.38
CCR2 P41597 1/20 0.37
NPC1 O15118 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C19 P33261 2/20 0.37
MTOR P42345 2/20 0.37
RAB9A P51151 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10102 0.88 ALDH1A1 (0.41) SLC7A5SLC6A9TRPM8NPC1RAB9A
SCHEMBL3486 0.88 TRPM8 (0.42) SLC7A5SLC6A9TRPM8NPC1RAB9A
SCHEMBL10451 0.87 PPARG (0.39) SLC7A5SLC6A9TRPM8PPARGPPARA
SCHEMBL7318201 0.83 SLC6A9 (0.60) SLC7A5SLC6A9SLC6A4HRH3NPC1
SCHEMBL10359727 0.83 SLC7A5 (0.52) SLC7A5SLC6A9SLC6A4HRH3TRPM8
SCHEMBL4660 0.82 HTR1A (0.46) SLC6A9SLC6A4HRH3CCR2NPC1
SCHEMBL3802 0.81 OPRM1 (0.48) SLC6A9SLC6A4HRH3PPARGPPARA
SCHEMBL4740321 0.80 SLC6A9 (0.57) SLC6A9SLC6A4HRH3NPC1CYP2D6
SCHEMBL4028 0.80 SLC6A4 (0.42) SLC6A4FFAR1CCR2NPC1CYP2D6
Oxalic Acid SCHEMBL10359897 0.77 SLC6A4 (0.62) SLC7A5SLC6A9SLC6A4HRH3CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5023269-A 3-aryloxy-3-substituted propanamines ELI LILLY AND COMPANY (US) 1991-06-11 US disclosed
EP-0273658-B1 3-ARYLOXY-3-SUBSTITUTED PROPANAMINES ELI LILLY AND COMPANY (US) 1990-10-31 EP disclosed
EP-0273658-A1 3-Aryloxy-3-substituted propanamines ELI LILLY AND COMPANY (US) 1988-07-06 EP disclosed