SCHEMBL10569739

SCHEMBL10569739

CC(=O)NC(=O)c1cncn1Cc1c(F)cccc1F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 5/20 0.38
PDE4A P27815 5/20 0.38
CYP11B1 P15538 2/20 0.37
CYP11B2 P19099 2/20 0.37
STIM1 Q13586 1/20 0.36
ORAI1 Q96D31 1/20 0.36
CA5A P35218 1/20 0.35
GPBAR1 Q8TDU6 2/20 0.35
KLKB1 P03952 4/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714132 0.87 GAA (0.40) PDE7APDE4ACYP11B1CYP11B2STIM1
SCHEMBL9714161 0.80 CA5A (0.48) PDE7APDE4ACYP11B1CYP11B2CA5A
SCHEMBL10564954 0.77 CYP11B2 (0.48) CYP11B1CYP11B2KDM4EALDH1A1
SCHEMBL10773961 0.72 ROCK2 (0.37) PDE7APDE4ACYP11B1CYP11B2CA5A
SCHEMBL9714339 0.72 RIPK1 (0.41) PDE7APDE4ACA5AKLKB1
SCHEMBL9857936 0.69 CA5A (0.66) CA5AKLKB1ALDH1A1
SCHEMBL9714409 0.66 AURKA (0.40) CA5AGPBAR1
SCHEMBL13328951 0.65 CES2 (0.52) ALDH1A1
SCHEMBL10569749 0.64 CYP11B2 (0.46) CYP11B1CYP11B2KDM4EALDH1A1
SCHEMBL9733613 0.64 GRK2 (0.36) CA5AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4851424-A 1-Phenyl-lower alkyl-imidazole 4- or 5-carboxamide compounds which are useful in the treatment of epilepsy CIBA-GEIGY CORPORATION (US) 1989-07-25 US disclosed