SCHEMBL10680751

SCHEMBL10680751

C[Si](C)(C)CCOC(=O)C(Br)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.47
CES1 P23141 2/20 0.47
CHRM1 P11229 6/20 0.43
CHRM3 P20309 5/20 0.43
CHRM2 P08172 4/20 0.43
CHRM4 P08173 4/20 0.43
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681761 0.83 ALDH1A1 (0.38) CYP1A2ALDH1A1SMN1; SMN2KMT2A
SCHEMBL2419442 0.81 LMNA (0.53) CES2CES1CHRM1CHRM3CHRM2
SCHEMBL28626716 0.81 SMN1; SMN2 (0.41) CES2CES1CHRM1CHRM3CHRM2
SCHEMBL2418494 0.80 TSHR (0.51) CES2CES1CHRM1CHRM3CHRM2
SCHEMBL28626193 0.80 NPC1 (0.42) CES2CES1CHRM1CHRM3CHRM2
SCHEMBL19086397 0.80 CES2 (0.53) CES2CES1CHRM1CHRM3CHRM2
SCHEMBL2417875 0.79 TSHR (0.53) CES2CES1CHRM1CHRM3CHRM2
SCHEMBL13523009 0.78 MTNR1A (0.55) CES2CES1ALDH1A1HPGD
SCHEMBL280401 0.78 MMP8 (0.56) CES2CES1SMN1; SMN2KMT2A
SCHEMBL26785147 0.77 CES2 (0.47) CES2CES1CHRM1CHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4794108-A BACTERICIDES, MICROBIOCIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-12-27 US disclosed
EP-0135194-A1 Azetidinones and their production Takeda Chemical Industries, Ltd. (JP) 1985-03-27 EP disclosed