SCHEMBL9681761

SCHEMBL9681761

COc1ccc(C(Br)C(=O)OCC[Si](C)(C)C)cc1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
GSK3B P49841 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
CYP1A2 P05177 1/20 0.38
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
MEN1 O00255 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9683539 0.84 GLS (0.41) ALDH1A1L3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL9683532 0.84 GLS (0.41) ALDH1A1L3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL10680751 0.83 CES2 (0.47) ALDH1A1KMT2ASMN1; SMN2CYP1A2
SCHEMBL6787347 0.80 ALOX15 (0.49) ALDH1A1KMT2AL3MBTL1GSK3BNPC1
SCHEMBL9683501 0.78 MTNR1A (0.38) ALDH1A1L3MBTL1NPC1RAB9ASMN1; SMN2
SCHEMBL378101 0.77 KMT2A (0.49) ALDH1A1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL1394924 0.75 PTGS2 (0.63) L3MBTL1CYP1A2
SCHEMBL1394923 0.75 PTGS2 (0.63) L3MBTL1CYP1A2
SCHEMBL9681759 0.75 TDP1 (0.41) ALDH1A1KMT2AL3MBTL1NPC1RAB9A
SCHEMBL8933321 0.72 ALDH1A1 (0.47) ALDH1A1KMT2AL3MBTL1GSK3BRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5087631-A Vasodilators for treating cardiovascular disorders GLAXO INC. (US) 1992-02-11 US disclosed