SCHEMBL10691683

SCHEMBL10691683

CCOC(=O)COc1ccc2c(c1)C(c1ccccc1)=NCc1ncc(C)n1-2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.44
KDM4E B2RXH2 4/20 0.44
MAPT P10636 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HSD17B10 Q99714 3/20 0.44
TP53 P04637 1/20 0.44
GABRA5 P31644 5/20 0.43
GABRA2 P47869 5/20 0.43
GABRA1 P14867 4/20 0.43
GAA P10253 3/20 0.43
GABRA3 P34903 2/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
GABRA4 P48169 1/20 0.43
GABRA6 Q16445 1/20 0.43
GABRB2 P47870 4/20 0.42
OPRK1 P41145 2/20 0.42
BRD4 O60885 1/20 0.42
LMNA P02545 1/20 0.42
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10694252 0.87 GABRA1 (0.58) HPGDKDM4EMAPTALDH1A1HSD17B10
SCHEMBL10691138 0.82 GABRA1 (0.49) HPGDALDH1A1GABRA5GABRA2GABRA1
SCHEMBL8933539 0.78 GABRA1 (0.47) HPGDKDM4EALDH1A1GABRA5GABRA2
SCHEMBL10694413 0.76 MAPK1 (0.45) ALDH1A1LMNA
SCHEMBL10692488 0.76 GABRA1 (0.62) HPGDALDH1A1GABRA5GABRA2GABRA1
SCHEMBL11809246 0.76 OPRK1 (0.69) HPGDKDM4ETP53GABRA5GABRA2
SCHEMBL11832211 0.76 GABRA5 (0.51) HPGDGABRA5GABRA2GABRA1GABRA3
SCHEMBL11826946 0.76 GABRA1 (0.69) HPGDKDM4EALDH1A1GABRA5GABRA2
SCHEMBL11835751 0.74 GABRA1 (0.49) HPGDGABRA5GABRA2GABRA1GABRA3
SCHEMBL11837344 0.73 LMNA (0.62) HPGDMAPTGABRA5GABRA2GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255028-A2 1,4-Benzodiazepines, their preparation and use as PAF antagonists BOEHRINGER INGELHEIM KG (DE) 1988-02-03 EP disclosed