SCHEMBL10692555

SCHEMBL10692555

COc1cc(S(N)(=O)=O)ccc1-c1nc2[nH]c(=O)ncc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 7/20 0.43
CA9 Q16790 7/20 0.43
CA12 O43570 6/20 0.43
CA1 P00915 6/20 0.43
CA4 P22748 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
PDE2A O00408 1/20 0.38
PDE5A O76074 2/20 0.38
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDR P35968 2/20 0.36
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10690895 0.88 TAS2R14 (0.40) KDM4EALDH1A1HPGDPDE2APDE5A
SCHEMBL10692548 0.87 MAPT (0.46) KDM4EALDH1A1HPGDPDE2APDE5A
SCHEMBL10691571 0.81 PDE2A (0.41) KDM4EALDH1A1HPGDPDE2APDE5A
SCHEMBL10689310 0.80 MKNK1 (0.47) EGFR
SCHEMBL10686293 0.79 GRIN2D (0.42) KDM4EALDH1A1HPGDPDE2APDE5A
SCHEMBL10690686 0.79 EGLN2 (0.39) KDM4EALDH1A1HPGDPDE2APDE5A
SCHEMBL10678075 0.78 PDE5A (0.49) CA2CA9CA12CA1CA4
SCHEMBL10744912 0.78 PDE2A (0.46) CA2CA9CA12CA1CA4
SCHEMBL10691563 0.77 CA2 (0.42) CA2CA9CA12CA1CA4
SCHEMBL10690657 0.76 CYP3A4 (0.49) CA2CA9CA12CA1CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722929-A Novel 2-phenyl-imidazoles and pharmaceutical compositions containing same DR. KARL THOMAE GMBH (DE) 1988-02-02 US disclosed
EP-0149200-A1 Novel 2-pnenyl-imidazoles, their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1985-07-24 EP disclosed