SCHEMBL10694088

SCHEMBL10694088

S=C([S-])NC1CCCCC1.[Na+]

nearest known ligand 0.61

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 known ✓ O43570 1/20 0.45
CA1 known ✓ P00915 1/20 0.45
CA2 known ✓ P00918 1/20 0.45
ALDH1A1 P00352 2/20 0.61
CYP3A4 P08684 2/20 0.61
TP53 P04637 1/20 0.61
SMN1; SMN2 Q16637 5/20 0.54
LMNA P02545 1/20 0.52
GAA P10253 1/20 0.52
NPC1 O15118 4/20 0.50
RAB9A P51151 3/20 0.50
MAPK1 P28482 1/20 0.50
DUSP3 P51452 1/20 0.50
PTPN5 P54829 1/20 0.50
PTPN11 Q06124 1/20 0.50
EPHX1 P07099 5/20 0.48
MAPT P10636 3/20 0.48
KDM4E B2RXH2 2/20 0.48
EPHX2 P34913 1/20 0.48
NPSR1 Q6W5P4 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28362407 0.97 SMN1; SMN2 (0.56) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL11483981 0.95 ALDH1A1 (0.61) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
Zinc Ion SCHEMBL28430295 0.92 SMN1; SMN2 (0.56) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL17670565 0.87 SMN1; SMN2 (0.48) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL3075946 0.76 ALDH1A1 (0.70) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL11842060 0.76 ALDH1A1 (1.00) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL491492 0.76 ALDH1A1 (1.00) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL11597254 0.76 ALDH1A1 (1.00) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL5695564 0.74 ALDH1A1 (0.67) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA
SCHEMBL24531349 0.72 ALDH1A1 (0.64) ALDH1A1CYP3A4TP53SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1087629-C Brain perfusion developer99mTcN(CHDT)2And method for preparing the same INST OF APPLIED CHEMISTRY BEIJ (CN) 2002-07-17 CN disclosed
CN-1280013-A Brain perfusion developer 99m TCN (CHDT)2 and its preparing method INST OF APPLIED CHEMISTRY BEIJ (CN) 2001-01-17 CN disclosed
EP-0266552-A1 Process for production of isothiocyanates STAUFFER CHEMICAL COMPANY (US) 1988-05-11 EP disclosed
US-4713467-A OXIDATION OF DITHIOCARBAMATES; METAL CATALYST; H CONTROL STAUFFER CHEMICAL COMPANY (US) 1987-12-15 US disclosed