SCHEMBL11021741

SCHEMBL11021741

CCOc1cc(S(=O)(=O)N(C)C)ccc1-c1nc2ccc(C#N)cc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.44
MAPT P10636 3/20 0.43
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
METAP2 P50579 1/20 0.42
METAP1 P53582 1/20 0.42
PKN1 Q16512 1/20 0.42
PKN2 Q16513 1/20 0.42
SRPK2 P78362 1/20 0.41
SRPK1 Q96SB4 1/20 0.41
CHEK2 O96017 1/20 0.40
TRPV4 Q9HBA0 1/20 0.39
CYP3A4 P08684 5/20 0.39
CYP2C9 P11712 5/20 0.39
CYP1A2 P05177 4/20 0.39
CYP2C19 P33261 4/20 0.39
CYP2D6 P10635 3/20 0.39
OGT O15294 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11021736 0.92 MAPT (0.43) ATRMAPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL11022217 0.89 ATR (0.53) ATRMAPTMETAP2METAP1PKN1
SCHEMBL11018866 0.89 MAPT (0.44) ATRMAPTALDH1A1SMN1; SMN2METAP2
SCHEMBL11021091 0.88 ATR (0.48) ATRMAPTALDH1A1SMN1; SMN2METAP2
SCHEMBL11021240 0.86 MAPT (0.46) ATRMAPTALDH1A1SMN1; SMN2METAP2
SCHEMBL11018857 0.81 MAPT (0.44) ATRMAPTALDH1A1MEN1LMNA
SCHEMBL11022213 0.81 ATR (0.44) ATRMAPTTRPV4PDE5A
SCHEMBL11021561 0.81 L3MBTL1 (0.47) ATRMAPTALDH1A1SMN1; SMN2METAP2
SCHEMBL11021081 0.80 CA12 (0.43) ATRMAPTCHEK2TRPV4KMT2A
SCHEMBL11018186 0.80 CYP3A4 (0.48) ATRPKN1PKN2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed