SCHEMBL11057576

SCHEMBL11057576

Cc1cccc(C(C)C)c1-n1cnc(N)nc1=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
HCAR1 Q9BXC0 2/20 0.38
ANPEP P15144 4/20 0.37
P2RX3 P56373 1/20 0.35
P2RX2 Q9UBL9 1/20 0.35
DPP4 P27487 5/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
DHFR P00374 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052581 0.87 HCAR1 (0.48) ALDH1A1HCAR1ANPEPDPP4
SCHEMBL11059558 0.85 FGFR1 (0.38) ALDH1A1HCAR1ANPEPP2RX3P2RX2
SCHEMBL11059375 0.81 HCAR1 (0.40) HCAR1ANPEPDPP4
SCHEMBL11054591 0.81 CHRNA7 (0.46) HCAR1
SCHEMBL11056242 0.81 HCAR1 (0.40) HCAR1ANPEPDPP4DHFR
SCHEMBL11054450 0.81 HCAR1 (0.40) HCAR1DPP4
SCHEMBL11056476 0.81 HCAR1 (0.40) ALDH1A1HCAR1ANPEPDPP4
SCHEMBL11054891 0.79 PKM (0.41) ALDH1A1HCAR1DHFR
SCHEMBL11057681 0.78 APLNR (0.39) ALDH1A1ALOX15TSHRHCAR1
SCHEMBL11060075 0.77 HCAR1 (0.37) ALDH1A1HCAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed