SCHEMBL11080480

SCHEMBL11080480

COc1ccccc1OCCN(Cc1ccccc1)CC(O)COc1cccc([N+](=O)[O-])c1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.50
ALDH1A1 P00352 5/20 0.46
TSHR P16473 2/20 0.46
HTR1A P08908 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
KDM4E B2RXH2 2/20 0.41
MAPT P10636 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 2/20 0.39
AGTR1 P30556 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11166442 0.85 POLB (0.47) POLBALDH1A1TSHRHTR1AADRA1D
SCHEMBL11078576 0.84 POLB (0.46) POLBALDH1A1TSHRHTR1AADRA1D
SCHEMBL11080474 0.78 HTR1A (0.43) POLBALDH1A1HTR1AADRA1DADRA1A
SCHEMBL7952028 0.76 L3MBTL1 (0.46) POLBALDH1A1TSHRKDM4EMAPT
SCHEMBL7952030 0.76 L3MBTL1 (0.46) POLBALDH1A1TSHRKDM4EMAPT
SCHEMBL11077053 0.76 POLB (0.52) POLBALDH1A1TSHRKDM4EMAPT
SCHEMBL13916263 0.76 POLB (0.49) POLBALDH1A1TSHRHTR1AADRA1D
SCHEMBL5375723 0.75 ADRB2 (0.62) POLBALDH1A1TSHRHTR1AADRA1D
Methyl Alcohol SCHEMBL11168835 0.75 ALDH1A1 (0.53) POLBALDH1A1TSHRMAPTCYP1A2
SCHEMBL11548958 0.74 POLB (0.57) POLBALDH1A1TSHRKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4438116-A Quinoxalinyloxy-amino-propanol compounds with blood pressure lowering and β-blocking properties, their use and pharmaceutical compositions containing them BOEHRINGER MANNHEIM GMBH (DE) 1984-03-20 US disclosed
EP-0019918-B1 DERIVATIVES OF AMINO-PROPANOL, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Roche Diagnostics GmbH (DE) 1983-09-07 EP disclosed