SCHEMBL11240

SCHEMBL11240

CCCCC(=O)N1CCN(C)CC1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.62
GNAI3 P08754 6/20 0.60
GNAI1 P63096 6/20 0.60
GNAO1 P09471 5/20 0.60
KMT2A Q03164 4/20 0.60
MEN1 O00255 3/20 0.60
TDP1 Q9NUW8 2/20 0.60
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
ATM Q13315 1/20 0.50
NPC1 O15118 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
HTR1A P08908 1/20 0.47
GPR183 P32249 1/20 0.47
CYP1A2 P05177 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548026 0.94 L3MBTL1 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL4548016 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL8972364 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL8972105 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL8972071 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL31632756 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL8972852 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL3339374 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL8972731 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A
SCHEMBL8973186 0.92 GNAI3 (0.71) L3MBTL1GNAI3GNAI1GNAO1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260068886-A1 COMPOSITIONS AND METHODS FOR TARGETED INHIBITION AND DEGRADATION OF PROTEINS IN AN INSECT CELL OERTH BIO LLC (US) 2026-03-12 US disclosed
EP-4580405-A1 COMPOSITIONS AND METHODS FOR TARGETED INHIBITION AND DEGRADATION OF PROTEINS IN AN INSECT CELL Oerth Bio LLC (US) 2025-07-09 EP disclosed
CN-116375715-B Compound serving as non-covalent BTK kinase inhibitor and biological application thereof 中国药科大学 2025-04-04 CN disclosed
WO-2024050016-A9 COMPOSITIONS AND METHODS FOR TARGETED INHIBITION AND DEGRADATION OF PROTEINS IN AN INSECT CELL OERTH BIO LLC (US) 2025-04-03 WO disclosed
US-20240365736-A1 COMPOSITIONS AND METHODS FOR TARGETED DEGRADATION OF PROTEINS IN A PLANT CELL OERTH BIO LLC (US) 2024-11-07 US disclosed
EP-4395549-A1 COMPOSITIONS AND METHODS FOR TARGETED DEGRADATION OF PROTEINS IN A PLANT CELL Oerth Bio LLC (US) 2024-07-10 EP disclosed
WO-2024050016-A1 COMPOSITIONS AND METHODS FOR TARGETED INHIBITION AND DEGRADATION OF PROTEINS IN AN INSECT CELL OERTH BIO LLC (US) 2024-03-07 WO disclosed
WO-2023034411-A1 COMPOSITIONS AND METHODS FOR TARGETED DEGRADATION OF PROTEINS IN A PLANT CELL OERTH BIO LLC (US) 2023-03-09 WO disclosed
EP-3728235-B1 SUBSTITUTED THIOPHENYLURACILS , THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS SYNGENTA CROP PROTECTION AG (CH) 2022-02-09 EP disclosed
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
US-20130281664-A1 NOVEL RUTHENIUM COMPLEXES AND THEIR USES IN PROCESSES FOR FORMATION AND/OR HYDROGENATION OF ESTERS, AMIDES AND DERIVATIVES THEREOF YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2013-10-24 US disclosed
US-20130190284-A1 X-Ray and Gamma-Photon Activable Organic Compounds, Their Preparation and Their Uses UNIVERSITE RENE PARIS DESCARTES (FR) 2013-07-25 US disclosed
WO-2013060860-A1 N-ACYL-N'-PHENYLPIPERAZINE DERIVATIVES AS SRBP MODULATORS FOR USE IN THE TREATMENT OF DIABETES AND OBESITY NATIONAL UNIVERSITY OF IRELAND, MAYNOOTH (IE) 2013-05-02 WO disclosed
US-20120253042-A1 USE OF RUTHENIUM COMPLEXES FOR FORMATION AND/OR HYDROGENATION OF AMIDES AND RELATED CARBOXYLIC ACID DERIVATIVES YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2012-10-04 US disclosed
US-20120253042-A1 USE OF RUTHENIUM COMPLEXES FOR FORMATION AND/OR HYDROGENATION OF AMIDES AND RELATED CARBOXYLIC ACID DERIVATIVES YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2012-10-04 US disclosed
WO-2012052996-A2 NOVEL RUTHENIUM COMPLEXES AND THEIR USES IN PROCESSES FOR FORMATION AND/OR HYDROGENATION OF ESTERS, AMIDES AND DERIVATIVES THEREOF YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2012-04-26 WO disclosed
WO-2012040204-A2 CYTOSOLIC FLUORESCENT ION INDICATORS ASANTE RESEARCH, LLC (US) 2012-03-29 WO disclosed
WO-2011048111-A1 COMPOUNDS RESPIVERT LIMITED (GB) 2011-04-28 WO disclosed
US-7560480-B2 Alkyl-containing 5-acylindolinones, the preparation thereof and their use as medicaments BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-07-14 US disclosed
US-7560480-B2 Alkyl-containing 5-acylindolinones, the preparation thereof and their use as medicaments BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120253042-A1 USE OF RUTHENIUM COMPLEXES FOR FORMATION AND/OR HYDROGENATION OF AMIDES AND RELATED CARBOXYLIC ACID DERIVATIVES ADH5, ADH1C, ADH1A L3MBTL1 4516/4885GNAI3 4150/4885GNAI1 4158/4885
US-20130190284-A1 X-Ray and Gamma-Photon Activable Organic Compounds, Their Preparation and Their Uses GLA, CGAS, VIP L3MBTL1 4320/4885GNAI3 218/4885GNAI1 177/4885
US-20240365736-A1 COMPOSITIONS AND METHODS FOR TARGETED DEGRADATION OF PROTEINS IN A PLANT CELL CRBN, LTN1, CBL L3MBTL1 157/4885GNAI3 3353/4885GNAI1 3222/4885
US-20130281664-A1 NOVEL RUTHENIUM COMPLEXES AND THEIR USES IN PROCESSES FOR FORMATION AND/OR HYDROGENATION OF ESTERS, AMIDES AND DERIVATIVES THEREOF ADH5, ADH1C, ADH1A L3MBTL1 4198/4885GNAI3 4353/4885GNAI1 4462/4885
US-20260068886-A1 COMPOSITIONS AND METHODS FOR TARGETED INHIBITION AND DEGRADATION OF PROTEINS IN AN INSECT CELL CRBN, STUB1, CUL1 L3MBTL1 191/4885GNAI3 2003/4885GNAI1 1959/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.