SCHEMBL1126650

SCHEMBL1126650

CCCc1cc(-c2ccccc2)c(C(=O)C(=O)Cl)n1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.41
PPARG P37231 1/20 0.40
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
HPGD P15428 2/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TSHR P16473 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127204 0.89 THRB (0.40) THRBALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL1126731 0.78 MMP1 (0.41) THRBALDH1A1HSD17B10SMN1; SMN2L3MBTL1
SCHEMBL15161896 0.76 CNR1 (0.38) THRBALDH1A1KDM4EHPGDLMNA
SCHEMBL15162096 0.75 THRB (0.39) THRBKDM4EHSD17B10SMN1; SMN2HPGD
SCHEMBL15162319 0.74 THRB (0.36) THRBALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL23488097 0.73 THRB (0.40) THRBALDH1A1KDM4ESMN1; SMN2HPGD
SCHEMBL1127235 0.72 THRB (0.37) THRBALDH1A1KDM4ESMN1; SMN2HPGD
SCHEMBL16500197 0.72 ALDH1A1 (0.44) ALDH1A1KDM4ESMN1; SMN2HPGDLMNA
SCHEMBL1993379 0.70 GABRA1 (0.40) THRBALDH1A1KDM4ESMN1; SMN2GAA
SCHEMBL1127116 0.70 LMNA (0.42) THRBALDH1A1KDM4ESMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-B1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2015-02-25 EP disclosed
EP-2626361-B1 Pyrrole antifungal agents F2G LTD (GB) 2014-10-15 EP disclosed
EP-2626361-A1 Pyrrole antifungal agents F2G Limited (GB) 2013-08-14 EP disclosed
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed