SCHEMBL1127186

SCHEMBL1127186

CC(=O)NCCc1c(C)[nH]c(C(=O)C(=O)Cl)c1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 11/20 0.45
MTNR1B P49286 10/20 0.45
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
HPGD P15428 2/20 0.43
CYP2C19 P33261 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP2D6 P10635 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
GFER P55789 1/20 0.42
MEN1 O00255 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1127399 0.81 LMNA (0.35) CYP1A2HPGDCYP2C19KDM4EALDH1A1
SCHEMBL1126894 0.79 LMNA (0.48) ALDH1A1TSHRNPC1LMNARAB9A
SCHEMBL1127778 0.79 LMNA (0.39) CYP1A2HPGDCYP2C19KDM4EALDH1A1
SCHEMBL1126936 0.79 CSF1R (0.39) CYP1A2CYP3A4CYP2C9HPGDCYP2C19
SCHEMBL1127408 0.74 RAB9A (0.39) CYP1A2HPGDCYP2C19KDM4EALDH1A1
SCHEMBL1126655 0.74 TBXAS1 (0.42) KDM4EALDH1A1TDP1RAB9ASMN1; SMN2
SCHEMBL1126902 0.73 LMNA (0.38) CYP1A2HPGDCYP2C19KDM4EALDH1A1
SCHEMBL1127366 0.72 LMNA (0.37) CYP1A2HPGDCYP2C19KDM4EALDH1A1
SCHEMBL1126974 0.71 LMNA (0.43) CYP1A2HPGDCYP2C19ALDH1A1TDP1
SCHEMBL1126648 0.69 CSF1R (0.37) CYP1A2HPGDCYP2C19KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2283006-A1 PYRROLE ANTIFUNGAL AGENTS F2G Limited (GB) 2011-02-16 EP disclosed
WO-2009130481-A1 PYRROLE ANTIFUNGAL AGENTS F2G LTD (GB) 2009-10-29 WO disclosed