SCHEMBL1128526

SCHEMBL1128526

CC(=O)Oc1ccc(S(C)(=O)=O)nc1C

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 15/20 0.43
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
RAB9A P51151 1/20 0.38
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16742542 0.82 KDM4E (0.39) KDM4EALDH1A1GAATSHRRAB9A
SCHEMBL16742902 0.77 MEN1 (0.54) KDM4EALDH1A1GAATSHRRAB9A
SCHEMBL2829068 0.74 GABRP (0.50) KDM4EALDH1A1GAATSHRRAB9A
SCHEMBL1128204 0.74 KDM4E (0.43) KDM4EALDH1A1GAATSHRRAB9A
SCHEMBL12813572 0.71 GPR119 (0.42) GPR119
SCHEMBL541733 0.71 ENPP2 (0.35) GPR119KDM4EALDH1A1GAA
SCHEMBL10133871 0.70 NOS3 (0.43) GPR119KDM4EALDH1A1GAAKMT2A
SCHEMBL10002447 0.69 NNMT (0.53) GPR119KDM4EALDH1A1
SCHEMBL2829457 0.69 ALDH1A1 (0.40) KDM4EALDH1A1GAATSHRRAB9A
SCHEMBL13458380 0.68 KDM4E (0.51) KDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188098-B2 GPR119 receptor agonists HOFFMANN-LA ROCHE INC. (US) 2012-05-29 US disclosed
CN-102036991-A GPR119 receptor agonists HOFFMANN LA ROCHE 2011-04-27 CN disclosed
EP-2283019-A1 GPR119 RECEPTOR AGONISTS F. Hoffmann-La Roche AG (CH) 2011-02-16 EP disclosed
WO-2009141238-A1 GPR119 RECEPTOR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-11-26 WO disclosed
US-20090286812-A1 GPR119 Receptor Agonists ERICKSON SHAWN DAVID 2009-11-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090286812-A1 GPR119 Receptor Agonists GPR119, GPR27, GPR139 GPR119 1/4885KDM4E 3907/4885ALDH1A1 973/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.