SCHEMBL11485145

SCHEMBL11485145

O=C([O-])C1(C(=O)[O-])CC(C(=O)[O-])(C(=O)[O-])C(C(=O)[O-])(C(=O)[O-])CC1(C(=O)[O-])C(=O)[O-].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+].[Na+]

nearest known ligand 0.38

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA4 known ✓ P22748 3/20 0.38
CA1 known ✓ P00915 1/20 0.35
FAHD1 Q6P587 1/20 0.38
MEN1 O00255 1/20 0.32
LDHA P00338 1/20 0.32
BLM P54132 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.30
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5886409 0.79 CA4 (0.38) CA4FAHD1CA1MEN1LDHA
SCHEMBL5886549 0.73 CA4 (0.33) CA4FAHD1CA1
SCHEMBL31220423 0.71 CA4 (0.38) CA4FAHD1CA1MEN1LDHA
Potassium Ion SCHEMBL16910245 0.71 CA4 (0.38) CA4FAHD1MEN1LDHABLM
SCHEMBL11580119 0.71 CA4 (0.32) CA4FAHD1CA1
SCHEMBL10918913 0.69 CA4 (0.30) CA4FAHD1
SCHEMBL30932964 0.67 CYP3A4 (0.39) CA4FAHD1CA1LMNA
Lithium Ion SCHEMBL5016617 0.67
Bicarbonate SCHEMBL29433967 0.66
Bicarbonate SCHEMBL16945860 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4182718-A BUILDERS, SQUESTRANTS, WATER SOFTENERS MONSANTO COMPANY (US) 1980-01-08 US disclosed
US-4107091-A COBALT, ALUMINUM AND ZINC OXIDES BATTELLE DEVELOPMENT CORPORATION (US) 1978-08-15 US disclosed
US-4092348-A Octasodium-1,1,2,2,4,4,5,5-cyclohexane octacarboxylate and compositions and methods employing same MONSANTO COMPANY (US) 1978-05-30 US disclosed
US-4092348-A Octasodium-1,1,2,2,4,4,5,5-cyclohexane octacarboxylate and compositions and methods employing same MONSANTO COMPANY (US) 1978-05-30 US disclosed
US-3997582-A Process and catalyst for synthesizing a gaseous hydrocarbon mixture having a high methane content from carbon monoxide and hydrogen BATTELLE DEVELOPMENT CORPORATION (US) 1976-12-14 US disclosed