SCHEMBL11526486

SCHEMBL11526486

Cc1c([N+]#N)cccc1C(F)(F)F.F[B-](F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 1/20 0.38
NOTUM Q6P988 1/20 0.34
CTSS P25774 1/20 0.34
AR P10275 1/20 0.33
DHODH Q02127 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HSD11B1 P28845 3/20 0.32
P2RX7 Q99572 1/20 0.31
CES1 P23141 1/20 0.31
ACHE P22303 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL260225 0.81 LMNA (0.36) ARHSD11B1
SCHEMBL13726323 0.77 TRPA1 (0.37) ACHE
SCHEMBL11523592 0.75 AR (0.37) TAS2R14ARHSD11B1P2RX7ACHE
SCHEMBL261312 0.74 ALDH1A1 (0.39) NOTUMARHSD11B1CES1
SCHEMBL4113607 0.74 ALDH1A1 (0.32)
SCHEMBL6630838 0.73 TAS2R14 (0.46) TAS2R14NOTUMCTSSDHODHHDAC6
SCHEMBL28772799 0.73 ALDH1A1 (0.31)
Hydrochloric Acid SCHEMBL18936435 0.72 ALDH1A1 (0.38) ARHSD11B1CES1
Hydrochloric Acid SCHEMBL9659775 0.72 ALDH1A1 (0.42) ARHSD11B1CES1
Fluoride Ion SCHEMBL11774111 0.72 ALDH1A1 (0.38) NOTUMARHSD11B1CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4132737-A ENZYME INHIBITORS ELI LILLY AND COMPANY (US) 1979-01-02 US disclosed