SCHEMBL11565347

SCHEMBL11565347

O=C(O)C(=Cc1ccccc1S)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.47
MAPT P10636 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
KDM4E B2RXH2 1/20 0.41
HTT P42858 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
AKR1C3 P42330 1/20 0.36
MDM4 O15151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16287426 0.84 TP53 (0.56) TP53KDM4EHTTCYP1A2CYP3A4
SCHEMBL11265544 0.77 MAPT (0.39) TP53MAPTKDM4E
SCHEMBL7607193 0.77 NFKB1 (0.53) TP53MAPTKDM4E
SCHEMBL5179024 0.76 TBXAS1 (0.40) MAPTHDAC8KDM4ECYP3A4CYP2C9
SCHEMBL7311482 0.75 TRPA1 (0.50) TP53MAPTHDAC8
SCHEMBL433478 0.75 TP53 (0.47) TP53MAPTKDM4EHTTCYP1A2
SCHEMBL7446722 0.75 ALDH1A1 (0.50) TP53MAPTKDM4EHTTCYP1A2
SCHEMBL8515208 0.72 TP53 (0.44) TP53MAPTKDM4EHTTCYP1A2
SCHEMBL7189395 0.72 KDM4E (0.71) TP53MAPTHDAC8KDM4EHTT
SCHEMBL11795578 0.72 CES2 (0.47) TP53MAPTHDAC8CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0003115-A1 Penicillins, per se and for use as antibacterially active antibiotics and their production SANDOZ AG (CH) 1979-07-25 EP disclosed