Risocaine

Risocaine

SCHEMBL118038

CCCOC(=O)c1ccc(N)cc1

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.80
CYP1A2 P05177 4/20 0.80
TSHR P16473 4/20 0.80
CYP3A4 P08684 3/20 0.80
CYP2C19 P33261 2/20 0.80
CYP2C9 P11712 1/20 0.80
PDE4D Q08499 1/20 0.80
ALDH1A1 P00352 4/20 0.75
RAB9A P51151 3/20 0.75
NPC1 O15118 2/20 0.75
MAPT P10636 1/20 0.75
MAOA P21397 2/20 0.72
ESR1 P03372 2/20 0.70
CHRM1 P11229 1/20 0.70
SLC6A2 P23975 1/20 0.70
KDR P35968 1/20 0.70
TDP1 Q9NUW8 1/20 0.70
CYP2D6 P10635 3/20 0.68
HTR3A P46098 1/20 0.68
HRH3 Q9Y5N1 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Risocaine SCHEMBL10481404 0.98 LMNA (0.77) LMNACYP1A2TSHRCYP3A4CYP2C19
Risocaine SCHEMBL21873190 0.98 LMNA (0.77) LMNACYP1A2TSHRCYP3A4CYP2C19
Risocaine SCHEMBL21647391 0.96 LMNA (0.75) LMNACYP1A2TSHRCYP3A4CYP2C19
SCHEMBL49950 0.90 ALDH1A1 (0.84) LMNACYP1A2TSHRCYP3A4CYP2C19
Butamben SCHEMBL81735 0.89 LMNA (1.00) LMNACYP1A2TSHRCYP3A4CYP2C19
SCHEMBL28758641 0.88 ALDH1A1 (0.81) LMNACYP1A2TSHRCYP3A4CYP2C19
SCHEMBL27647586 0.88 ALDH1A1 (0.81) LMNACYP1A2TSHRCYP3A4CYP2C19
SCHEMBL27667930 0.88 ALDH1A1 (0.81) LMNACYP1A2TSHRCYP3A4CYP2C19
SCHEMBL27647510 0.88 ALDH1A1 (0.81) LMNACYP1A2TSHRCYP3A4CYP2C19
SCHEMBL27667922 0.88 ALDH1A1 (0.81) LMNACYP1A2TSHRCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1812 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144801-A1 COMPOSITIONS AND METHODS FOR PREVENTING OR TREATING MUSCLE CONDITIONS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-05-28 US claimed
WO-2025235864-A1 COATED NEEDLE ADMINISTRATION SYSTEMS EVOLUS, INC. (US) 2025-11-13 WO claimed
EP-4578441-A1 TREATMENT OF LOCALIZED PAIN PlantTec Medical GmbH (DE) 2025-07-02 EP claimed
CN-119925187-A Oral care composition and method for maintaining oral hygiene using the same 进化牙白金有限公司 2025-05-06 CN claimed
WO-2025085689-A1 EXTRACELLULAR SMALL MOLECULE ACTIVATORS TARGETING BESTROPHIN CHANNELS FOR DISEASE TREATMENT THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2025-04-24 WO claimed
EP-3703802-B9 NASAL DELIVERY DEVICES AND METHODS OF USE THEREOF CLEXIO BIOSCIENCES LTD (IL) 2024-12-04 EP claimed
EP-3703802-B1 NASAL DELIVERY DEVICES AND METHODS OF USE THEREOF CLEXIO BIOSCIENCES LTD (IL) 2024-10-16 EP claimed
EP-3863708-B1 MIXED IONIC CONDUCTORS AND CORRESPONDING DEVICES, SYSTEMS AND METHODS OF MAKING BATTELLE MEMORIAL INSTITUTE (US) 2024-09-11 EP claimed
US-20240197867-A1 NEURAL CONTROL OF ADAPTIVE IMMUNITY THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH 2024-06-20 US claimed
US-20240165247-A1 NEW PEPTIDE CONJUGATES Enlitisa (Shanghai) Pharmaceutical Co., Ltd. (CN) 2024-05-23 US claimed
US-20010055607-A1 COMPOSITIONS, KITS, AND METHODS FOR INHIBITING CEREBRAL NEUROVASCULAR DISORDERS AND MUSCULAR HEADACHES BHL PATENT HOLDINGS LLC 2001-12-27 US claimed
US-20010004644-A1 Compositions, kits, apparatus, and methods for inhibiting cephalic inflammation LEVIN BRUCE H (US) 2001-06-21 US claimed
WO-2001043733-A2 COMPOSITIONS, KITS, APPARATUS, AND METHODS FOR INHIBITING CEPHALIC INFLAMMATION LEVIN BRUCE H (US) 2001-06-21 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
US-6207178-B1 STABLE SUSPENSION KABI PHARMACIA AB (SE) 2001-03-27 US claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-5785976-A Solid lipid particles, particles of bioactive agents and methods for the manufacture and use thereof PHARMACIA & UPJOHN AB (SE) 1998-07-28 US claimed
EP-0687172-A1 SOLID LIPID PARTICLES, PARTICLES OF BIOACTIVE AGENTS AND METHODS FOR THE MANUFACTURE AND USE THEREOF Pharmacia & Upjohn Aktiebolag (SE) 1995-12-20 EP claimed
WO-1994020072-A1 SOLID LIPID PARTICLES, PARTICLES OF BIOACTIVE AGENTS AND METHODS FOR THE MANUFACTURE AND USE THEREOF PHARMACIA AB (SE) 1994-09-15 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010055607-A1 COMPOSITIONS, KITS, AND METHODS FOR INHIBITING CEREBRAL NEUROVASCULAR DISORDERS AND MUSCULAR HEADACHES TNNC1, KIT, PDE3A LMNA 477/4885CYP1A2 2135/4885TSHR 4600/4885
US-20010004644-A1 Compositions, kits, apparatus, and methods for inhibiting cephalic inflammation CXCR5, CCL5, C5AR2 LMNA 1480/4885CYP1A2 1652/4885TSHR 4356/4885
US-20240197867-A1 NEURAL CONTROL OF ADAPTIVE IMMUNITY TRPV1, TRPA1, TRPV2 LMNA 4746/4885CYP1A2 4785/4885TSHR 3276/4885
US-20260144801-A1 COMPOSITIONS AND METHODS FOR PREVENTING OR TREATING MUSCLE CONDITIONS CPT1B, HPGD, PTGES LMNA 1427/4885CYP1A2 360/4885TSHR 2274/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.